SCHEMBL8562631

SCHEMBL8562631

CCOC(=O)CC(c1ccccc1)c1ccc(-n2ccn(-c3ccc4c(c3)CCN(C(=O)C(F)(F)F)CC4)c2=O)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 7/20 0.39
SIGMAR1 Q99720 7/20 0.39
SLC6A2 P23975 2/20 0.39
HRH2 P25021 2/20 0.39
HRH1 P35367 2/20 0.39
HTR1A P08908 1/20 0.39
CHRM5 P08912 1/20 0.39
ADRA1D P25100 1/20 0.39
HTR1B P28222 1/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
HTR1E P28566 1/20 0.39
HTR2B P41595 1/20 0.39
SLC6A3 Q01959 1/20 0.39
MTNR1B P49286 1/20 0.39
ESR1 P03372 3/20 0.37
ESR2 Q92731 3/20 0.37
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4682332 0.82 ESR1 (0.50) TMEM97SIGMAR1SLC6A2HRH2HRH1
SCHEMBL7472118 0.81 ESR1 (0.41) TMEM97SIGMAR1SLC6A2HRH2HRH1
SCHEMBL8562345 0.80 ESR1 (0.39) TMEM97SIGMAR1SLC6A2HRH2HRH1
SCHEMBL7472374 0.80 TMEM97 (0.43) TMEM97SIGMAR1SLC6A2HRH2HRH1
SCHEMBL8897664 0.74 KMT2A (0.37) MTNR1BESR1ESR2KDM4EALDH1A1
SCHEMBL8559513 0.73 MTNR1B (0.36) TMEM97SIGMAR1SLC6A2HRH2HRH1
SCHEMBL4680153 0.71 ESR1 (0.55) ESR1ESR2HRH3
SCHEMBL7560796 0.71 ESR1 (0.42) TMEM97SIGMAR1SLC6A2HRH2HRH1
SCHEMBL7474127 0.70 TMEM97 (0.43) TMEM97SIGMAR1SLC6A2HRH2HRH1
SCHEMBL8561816 0.69 ESR1 (0.36) TMEM97SIGMAR1SLC6A2HRH2HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0612741-B1 Cyclic derivatives, medicaments containing them and process for their preparation THOMAE GMBH DR K (DE) 1998-06-10 EP disclosed
US-5612335-A ANTICOAGULANTS; COMBATING/PREVENTING DISEASES WHERE CELL AGGREGATES OCCUR OR CELL-MATRIX INTERACTIONS PLAY A PART KARL THOMAE GMBH (DE) 1997-03-18 US disclosed
US-5519036-A IMIDAZOLIDINONES, ANTICOAGULANTS, CELL AGGREGATION PREVENTION KARL THOMAE GMBH (DE) 1996-05-21 US disclosed
EP-0612741-A1 Cyclic derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1994-08-31 EP disclosed