SCHEMBL7472374

SCHEMBL7472374

CCOC(=O)CCn1ccn(-c2ccc3c(c2)CCN(C(=O)C(F)(F)F)CC3)c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 7/20 0.43
SIGMAR1 Q99720 7/20 0.43
SLC6A2 P23975 2/20 0.43
HRH2 P25021 2/20 0.43
HRH1 P35367 2/20 0.43
HTR1A P08908 1/20 0.43
CHRM5 P08912 1/20 0.43
ADRA1D P25100 1/20 0.43
HTR1B P28222 1/20 0.43
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
HTR1E P28566 1/20 0.43
HTR2B P41595 1/20 0.43
SLC6A3 Q01959 1/20 0.43
ESR1 P03372 3/20 0.40
ESR2 Q92731 3/20 0.40
CHRM1 P11229 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
TNF P01375 1/20 0.36
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7472118 0.91 ESR1 (0.41) TMEM97SIGMAR1SLC6A2HRH2HRH1
SCHEMBL7474127 0.80 TMEM97 (0.43) TMEM97SIGMAR1SLC6A2HRH2HRH1
SCHEMBL8562631 0.80 TMEM97 (0.39) TMEM97SIGMAR1SLC6A2HRH2HRH1
SCHEMBL8566035 0.79 ESR1 (0.40) HRH1ESR1ESR2KDM4ESMN1; SMN2
SCHEMBL8562345 0.78 ESR1 (0.39) TMEM97SIGMAR1SLC6A2HRH2HRH1
SCHEMBL7560796 0.74 ESR1 (0.42) TMEM97SIGMAR1SLC6A2HRH2HRH1
SCHEMBL8562237 0.73 ESR1 (0.39) ESR1ESR2
SCHEMBL8562233 0.73 ESR1 (0.39) ESR1ESR2
SCHEMBL8564893 0.72 ESR1 (0.39) ESR1ESR2
SCHEMBL8564898 0.72 ESR1 (0.39) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0777667-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT Dr. Karl Thomae GmbH (DE) 1997-06-11 EP disclosed
WO-1996005194-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT DR. KARL THOMAE GMBH (DE) 1996-02-22 WO disclosed