SCHEMBL8562708

SCHEMBL8562708

Cc1ccsc1C(=O)N(C)c1ccc(C(=O)N2Cc3ccccc3Cc3ccccc32)cc1

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 9/20 0.50
AVPR2 P30518 8/20 0.50
RAB9A P51151 3/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
NPC1 O15118 2/20 0.40
HPGD P15428 1/20 0.40
KMT2A Q03164 1/20 0.40
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8555958 0.87 AVPR1A (0.49) AVPR1AAVPR2RAB9ASMN1; SMN2NPC1
SCHEMBL8561629 0.84 AVPR2 (0.52) AVPR1AAVPR2RAB9ASMN1; SMN2NPC1
SCHEMBL7340044 0.84 AVPR1A (0.60) AVPR1AAVPR2
SCHEMBL8561249 0.82 AVPR2 (0.50) AVPR1AAVPR2
SCHEMBL8558249 0.82 NPC1 (0.45) AVPR1AAVPR2RAB9ASMN1; SMN2NPC1
SCHEMBL8564119 0.82 AVPR2 (0.68) AVPR1AAVPR2KMT2A
SCHEMBL8559549 0.81 AVPR1A (0.42) AVPR1AAVPR2RAB9ASMN1; SMN2NPC1
SCHEMBL8562373 0.81 AVPR1A (0.45) AVPR1AAVPR2RAB9ASMN1; SMN2NPC1
SCHEMBL8561048 0.80 AVPR2 (0.48) AVPR1AAVPR2
SCHEMBL8563827 0.80 ALDH1A1 (0.47) AVPR1AAVPR2RAB9ASMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed