SCHEMBL8563069

SCHEMBL8563069

Cc1ccc2c(c1)CNc1ccccc1S2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 6/20 0.43
KMT2A Q03164 6/20 0.43
HTT P42858 2/20 0.43
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 1/20 0.43
HPGD P15428 1/20 0.43
ATM Q13315 1/20 0.43
NOX1 Q9Y5S8 10/20 0.41
GAA P10253 7/20 0.41
MAPT P10636 6/20 0.41
ALOX15 P16050 3/20 0.41
BCHE P06276 2/20 0.41
ACHE P22303 2/20 0.41
SNCA P37840 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
CYP1A2 P05177 1/20 0.41
POLB P06746 1/20 0.41
CYP3A4 P08684 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
ALOX12 P18054 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4510651 0.81 GAA (0.52) MEN1KMT2AALDH1A1KDM4EHPGD
SCHEMBL8558177 0.81 NOX1 (0.58) MEN1KMT2AHPGDNOX1GAA
SCHEMBL8558747 0.80 NOX1 (0.61) MEN1KMT2AHTTALDH1A1NOX1
SCHEMBL225829 0.74 NOX1 (0.65) MEN1KMT2AHTTALDH1A1NOX1
SCHEMBL4731236 0.74 ALDH1A1 (0.53) MEN1KMT2AHTTALDH1A1KDM4E
SCHEMBL125602 0.74 ALDH1A1 (0.61) MEN1KMT2AHTTALDH1A1KDM4E
SCHEMBL29829120 0.74 ALDH1A1 (0.61) MEN1KMT2AHTTALDH1A1KDM4E
SCHEMBL28639550 0.73 ALDH1A1 (0.59) MEN1KMT2AHTTALDH1A1KDM4E
SCHEMBL8562468 0.71 NOX1 (0.58) MEN1KMT2AHPGDNOX1GAA
SCHEMBL8561569 0.71 MEN1 (0.47) MEN1KMT2AALDH1A1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed
EP-0640592-A1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID COMPANY (US) 1995-03-01 EP disclosed