SCHEMBL8558747

SCHEMBL8558747

COc1ccc2c(c1)CNc1ccccc1S2

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOX1 Q9Y5S8 7/20 0.61
GAA P10253 4/20 0.57
MAPT P10636 4/20 0.57
MEN1 O00255 3/20 0.57
KMT2A Q03164 3/20 0.57
MAPK1 P28482 3/20 0.57
TDP1 Q9NUW8 2/20 0.57
HTT P42858 2/20 0.57
SMN1; SMN2 Q16637 2/20 0.57
LMNA P02545 2/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
RYR2 Q92736 3/20 0.48
KCNH2 Q12809 1/20 0.48
PDE3B Q13370 1/20 0.46
PDE3A Q14432 1/20 0.46
SNCA P37840 3/20 0.45
KDM1A O60341 1/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8563265 0.88 NOX1 (0.61) NOX1GAAMAPTMEN1KMT2A
SCHEMBL10671438 0.85 NOX1 (0.61) NOX1GAAMAPTMEN1KMT2A
SCHEMBL8563069 0.80 MEN1 (0.43) NOX1GAAMAPTMEN1KMT2A
SCHEMBL4510651 0.77 GAA (0.52) NOX1GAAMAPTMEN1KMT2A
SCHEMBL8558177 0.77 NOX1 (0.58) NOX1GAAMAPTMEN1KMT2A
Phenothiazine SCHEMBL9074312 0.76 NOX1 (1.00) NOX1GAAMAPTMEN1KMT2A
SCHEMBL29278502 0.76 NOX1 (0.53) NOX1GAAMAPTMEN1KMT2A
SCHEMBL29936312 0.76 NOX1 (0.53) NOX1GAAMAPTMEN1KMT2A
SCHEMBL239600 0.76 NOX1 (1.00) NOX1GAAMAPTMEN1KMT2A
Benzene SCHEMBL29242182 0.75 NOX1 (0.97) NOX1GAAMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed
EP-0640592-A1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID COMPANY (US) 1995-03-01 EP disclosed