SCHEMBL8563186

SCHEMBL8563186

CC(=O)Nc1cc(O)c(C(C)=O)cc1[N+](=O)[O-]

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.51
NPSR1 Q6W5P4 2/20 0.51
POLB P06746 3/20 0.51
SMN1; SMN2 Q16637 3/20 0.51
GALR2 O43603 1/20 0.51
MITF O75030 1/20 0.51
ALDH1A1 P00352 1/20 0.51
LMNA P02545 1/20 0.51
HSP90AA1 P07900 1/20 0.51
HPGD P15428 1/20 0.51
XBP1 P17861 1/20 0.51
CCR6 P51684 1/20 0.51
HTT P42858 2/20 0.49
KMT2A Q03164 2/20 0.46
SLC9A1 P19634 1/20 0.44
PKM P14618 2/20 0.43
KCNMA1 Q12791 3/20 0.43
ALDH3A1 P30838 1/20 0.42
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2129921 0.89 NPSR1 (0.50) MAPTNPSR1POLBSMN1; SMN2GALR2
SCHEMBL2128713 0.87 SMN1; SMN2 (0.54) MAPTNPSR1POLBSMN1; SMN2GALR2
SCHEMBL27426629 0.85 RECQL (0.48) MAPTNPSR1POLBSMN1; SMN2GALR2
SCHEMBL29405447 0.83 NPSR1 (0.50) MAPTNPSR1POLBSMN1; SMN2GALR2
SCHEMBL21989034 0.83 SLC9A1 (0.52) MAPTNPSR1POLBSMN1; SMN2GALR2
SCHEMBL11095126 0.83 MAPT (0.52) MAPTNPSR1POLBSMN1; SMN2GALR2
SCHEMBL8767277 0.81 MAPT (0.51) MAPTNPSR1POLBSMN1; SMN2GALR2
SCHEMBL11951437 0.81 ALDH1A1 (0.51) MAPTNPSR1POLBSMN1; SMN2GALR2
SCHEMBL13811009 0.79 NPSR1 (0.49) MAPTNPSR1POLBSMN1; SMN2GALR2
SCHEMBL8954112 0.78 SMN1; SMN2 (0.58) MAPTNPSR1POLBSMN1; SMN2GALR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431943-B1 Spiro(pyran)piperidine derivatives MERCK & CO INC (US) 1998-07-15 EP disclosed
US-5633247-A ANTIARRTHYMIA AGENT MERCK & CO., INC. (US) 1997-05-27 US disclosed
CN-1110685-A Nitrogen-containing spiro ring MERCK & CO INC (US) 1995-10-25 CN disclosed
US-5206240-A Antiarrhythmia agents MERCK & CO., INC. (US) 1993-04-27 US disclosed
CN-1053613-A Nitrogen-containing spiro ring MERCK & CO INC (US) 1991-08-07 CN disclosed
EP-0431943-A2 Nitrogen-containing spirocycles MERCK & CO. INC. (US) 1991-06-12 EP disclosed