SCHEMBL8563265

SCHEMBL8563265

COc1ccc2c(c1)NCc1ccccc1S2

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOX1 Q9Y5S8 3/20 0.61
LMNA P02545 3/20 0.54
MAPT P10636 2/20 0.54
MAPK1 P28482 2/20 0.54
MEN1 O00255 1/20 0.54
GAA P10253 1/20 0.54
HTT P42858 1/20 0.54
KMT2A Q03164 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
SNCA P37840 2/20 0.45
PDE3B Q13370 1/20 0.42
PDE3A Q14432 1/20 0.42
RYR2 Q92736 2/20 0.41
KCNH2 Q12809 2/20 0.41
KDM1A O60341 1/20 0.38
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
CYP1A2 P05177 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10671438 0.88 NOX1 (0.61) NOX1LMNAMAPTMAPK1MEN1
SCHEMBL8558747 0.88 NOX1 (0.61) NOX1LMNAMAPTMAPK1MEN1
SCHEMBL4510651 0.77 GAA (0.52) NOX1MAPTMAPK1MEN1GAA
SCHEMBL8562468 0.77 NOX1 (0.58) NOX1LMNAMAPTMAPK1MEN1
Phenothiazine SCHEMBL9074312 0.76 NOX1 (1.00) NOX1LMNAMAPTMAPK1MEN1
SCHEMBL29936312 0.76 NOX1 (0.53) NOX1LMNAMAPTMAPK1MEN1
SCHEMBL29278502 0.76 NOX1 (0.53) NOX1LMNAMAPTMAPK1MEN1
SCHEMBL239600 0.76 NOX1 (1.00) NOX1LMNAMAPTMAPK1MEN1
Benzene SCHEMBL29242182 0.75 NOX1 (0.97) NOX1LMNAMAPTMAPK1MEN1
SCHEMBL25414339 0.74 PDE3B (0.45) NOX1LMNAMAPTMAPK1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed
EP-0640592-A1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID COMPANY (US) 1995-03-01 EP disclosed