SCHEMBL8563337

SCHEMBL8563337

O=C(Cc1ccccc1Cl)Nc1ccc(C(=O)N2Cc3ccccc3Cc3cc(Cl)ccc32)cc1

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 4/20 0.51
AVPR1A P37288 4/20 0.51
KCNJ5 P48544 3/20 0.48
KCNJ3 P48549 3/20 0.48
HSD17B3 P37058 1/20 0.43
THRB P10828 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8556372 0.91 KCNJ5 (0.51) AVPR2AVPR1AKCNJ5KCNJ3THRB
SCHEMBL8561770 0.91 AVPR2 (0.47) AVPR2AVPR1AHSD17B3
SCHEMBL8560236 0.88 MEN1 (0.48) AVPR2AVPR1A
SCHEMBL8559196 0.85 THRB (0.55) KCNJ5KCNJ3THRB
SCHEMBL8561962 0.83 AVPR2 (0.58) AVPR2AVPR1A
SCHEMBL8556841 0.83 AVPR2 (0.65) AVPR2AVPR1A
SCHEMBL8562554 0.82 AVPR2 (0.73) AVPR2AVPR1A
SCHEMBL8559571 0.82 AVPR2 (0.62) AVPR2AVPR1A
SCHEMBL8558803 0.81 NAMPT (0.57) AVPR2AVPR1A
SCHEMBL7340964 0.81 KCNJ5 (0.48) KCNJ5KCNJ3THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed