SCHEMBL8563536

SCHEMBL8563536

CS(=O)(=O)[N+]1(NC(=O)C(COCc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC2(CCNCC2)c2ccccc21

nearest known ligand 0.45

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 17/20 0.45
CYP3A4 P08684 1/20 0.37
UGCG Q16739 1/20 0.37
GHSR Q92847 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8561651 0.95 TACR1 (0.42) TACR1GHSR
SCHEMBL8564711 0.93 TACR1 (0.43) TACR1CYP3A4UGCGGHSR
SCHEMBL8566409 0.92 TACR1 (0.53) TACR1
SCHEMBL8562851 0.92 TACR1 (0.43) TACR1CYP3A4UGCG
SCHEMBL8560379 0.91 CTSL (0.40) TACR1UGCGGHSR
SCHEMBL8559045 0.90 TACR1 (0.41) TACR1CYP3A4UGCG
SCHEMBL8560138 0.90 TACR1 (0.41) TACR1CYP3A4UGCG
SCHEMBL8559389 0.90 TACR1 (0.42) TACR1GHSR
SCHEMBL8559555 0.90 TACR1 (0.40) TACR1GHSR
SCHEMBL8561114 0.90 TACR1 (0.40) TACR1CYP3A4UGCGGHSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5811431-A Spiro-substituted azacyclic derivatives and their use as therapeutic agents MERCK SHARP & DOHME LTD. (GB) 1998-09-22 US disclosed