SCHEMBL8563544

SCHEMBL8563544

O=[C]CN(NC(=O)c1cccnc1)C(=O)/C=C/c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
CYP1A1 P04798 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP1B1 Q16678 1/20 0.53
LMNA P02545 2/20 0.53
KDM4E B2RXH2 2/20 0.53
MAPT P10636 5/20 0.47
GAA P10253 1/20 0.47
HDAC1 Q13547 2/20 0.46
HDAC6 Q9UBN7 2/20 0.46
HDAC3 O15379 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC10 Q969S8 1/20 0.46
HDAC11 Q96DB2 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8563549 1.00 ALDH1A1 (0.56) ALDH1A1CYP2C9CYP2C19CYP1A1CYP1A2
SCHEMBL7750101 0.88 NPC1 (0.46) ALDH1A1CYP2C9CYP1A2CYP2D6CYP1B1
SCHEMBL7750096 0.88 NPC1 (0.46) ALDH1A1CYP2C9CYP1A2CYP2D6CYP1B1
SCHEMBL8566374 0.87 USP2 (0.45) ALDH1A1CYP2C9CYP2C19CYP1A1CYP1A2
SCHEMBL8566376 0.87 USP2 (0.45) ALDH1A1CYP2C9CYP2C19CYP1A1CYP1A2
SCHEMBL7746456 0.80 NPC1 (0.51) ALDH1A1CYP2C19CYP1A2LMNAKDM4E
SCHEMBL7746460 0.80 NPC1 (0.51) ALDH1A1CYP2C19CYP1A2LMNAKDM4E
SCHEMBL7749839 0.77 NPC1 (0.50) ALDH1A1CYP2C9CYP1A2CYP2D6CYP1B1
SCHEMBL7749846 0.77 NPC1 (0.50) ALDH1A1CYP2C9CYP1A2CYP2D6CYP1B1
SCHEMBL7747853 0.77 NPC1 (0.47) ALDH1A1CYP2C9CYP1A2CYP2D6CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0596406-B1 Imidazo (1,2-a) Pyridines as bradykinin antagonists FUJISAWA PHARMACEUTICAL CO (JP) 1998-12-16 EP disclosed
EP-0596406-A1 Imidazo (1,2-a) Pyridines as bradykinin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-05-11 EP disclosed