Bromide

Bromide

SCHEMBL8563893

O=C1C([P+](c2ccccc2)(c2ccccc2)c2ccccc2)CCN1Cc1ccc(C(F)(F)F)cc1.[Br-]

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHKACHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGHRH2OPRM1

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACHE known ✓ P22303 2/20 0.43
BCHE P06276 2/20 0.43
BACE1 P56817 2/20 0.43
SIGMAR1 Q99720 3/20 0.42
TEAD1 P28347 1/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
KCNH2 Q12809 1/20 0.41
CLPP Q16740 1/20 0.41
SIRT2 Q8IXJ6 1/20 0.40
SIRT1 Q96EB6 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL8900165 1.00 BCHE (0.43) BCHEACHEBACE1SIGMAR1TEAD1
Bromide SCHEMBL8563395 0.87 HDAC1 (0.43) ALDH1A1
Bromide SCHEMBL8563399 0.87 HDAC1 (0.43) ALDH1A1
Bromide SCHEMBL8900117 0.86 KCNH2 (0.44) ALDH1A1KCNH2
Bromide SCHEMBL8559098 0.86 KCNH2 (0.44) ALDH1A1KCNH2
Bromide SCHEMBL8480945 0.84 CYP3A4 (0.41) SIGMAR1KDM4EALDH1A1CLPP
Bromide SCHEMBL8478935 0.84 CYP3A4 (0.41) SIGMAR1KDM4EALDH1A1CLPP
Bromide SCHEMBL8567147 0.81 SIGMAR1 (0.47) SIGMAR1
Bromide SCHEMBL8899316 0.81 SIGMAR1 (0.47) SIGMAR1
Bromide SCHEMBL7887318 0.80 BCHE (0.46) BCHEACHEBACE1SIGMAR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5804577-A ANTIBIOTICS HOFFMANN-LA ROCHE INC. (US) 1998-09-08 US disclosed
EP-0761673-A1 Cephalosporin derivatives F. HOFFMANN-LA ROCHE AG (CH) 1997-03-12 EP disclosed