SCHEMBL8563978

SCHEMBL8563978

COc1cc(CNc2c([AsH]C(C)(C)C)c(=O)c2=O)cc(OC)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 1/20 0.39
TSHR P16473 3/20 0.37
ALDH1A1 P00352 2/20 0.37
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
ABCB1 P08183 1/20 0.36
ROCK2 O75116 1/20 0.34
GSK3A P49840 1/20 0.34
GSK3B P49841 1/20 0.34
ROCK1 Q13464 1/20 0.34
PRKG1 Q13976 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
TACR1 P25103 1/20 0.34
DHFR P00374 1/20 0.34
AURKA O14965 1/20 0.34
RPS6KB1 P23443 1/20 0.34
AURKB Q96GD4 1/20 0.34
KDM4E B2RXH2 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7895077 0.79 HIF1A (0.41) HIF1ATSHRALDH1A1MEN1KMT2A
SCHEMBL8569067 0.70 CHEK2 (0.32) ROCK2GSK3AGSK3BROCK1PRKG1
SCHEMBL12933384 0.66 TSHR (0.49) HIF1ATSHRALDH1A1MEN1KMT2A
SCHEMBL19325340 0.63 MEN1 (0.47) TSHRALDH1A1MEN1KMT2AL3MBTL1
SCHEMBL7887076 0.63 GSK3A (0.43) TSHRALDH1A1MEN1KMT2AROCK2
SCHEMBL5545073 0.63 HIF1A (0.55) HIF1ATSHRALDH1A1MEN1KMT2A
SCHEMBL681502 0.63 ALDH1A1 (0.53) HIF1ATSHRALDH1A1MEN1KMT2A
SCHEMBL8436952 0.61 CHRM2 (0.53) HIF1ATSHRALDH1A1MEN1KMT2A
SCHEMBL11619531 0.61 TSHR (0.52) HIF1ATSHRALDH1A1MEN1KMT2A
SCHEMBL27975799 0.61 CHEK1 (0.41) TSHRALDH1A1ROCK2GSK3AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934257-A1 SUBSTITUTED N-ARYLMETHYLAMINO DERIVATIVES OF CYCLOBUTENE-3,4-DIONES AMERICAN HOME PRODUCTS CORPORATION (US) 1999-08-11 EP disclosed
WO-1998002413-A1 SUBSTITUTED N-ARYLMETHYLAMINO DERIVATIVES OF CYCLOBUTENE-3,4-DIONES AMERICAN HOME PRODUCTS CORPORATION (US) 1998-01-22 WO disclosed