SCHEMBL8564220

SCHEMBL8564220

CCOC(=O)CCCc1ccccc1I

nearest known ligand 0.64

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 3/20 0.64
CYP4A11 Q02928 3/20 0.64
SMN1; SMN2 Q16637 2/20 0.60
CYP1A2 P05177 2/20 0.60
CYP3A4 P08684 1/20 0.60
CYP2D6 P10635 1/20 0.60
CYP2C9 P11712 1/20 0.60
CYP2C19 P33261 1/20 0.60
ALOX5 P09917 1/20 0.50
ALDH1A1 P00352 3/20 0.45
NAMPT P43490 1/20 0.44
GAA P10253 1/20 0.44
TOP2A P11388 1/20 0.43
CYP4Z1 Q86W10 1/20 0.43
CYP4F11 Q9HBI6 1/20 0.43
CYP4F12 Q9HCS2 1/20 0.43
TNF P01375 1/20 0.42
MAPT P10636 1/20 0.42
PKM P14618 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17284798 0.87 CYP4F2 (0.56) CYP4F2CYP4A11SMN1; SMN2CYP1A2CYP3A4
SCHEMBL12848923 0.85 CYP4F2 (0.47) CYP4F2CYP4A11SMN1; SMN2CYP1A2CYP3A4
SCHEMBL17244592 0.84 ALDH1A1 (0.52) CYP4F2CYP4A11SMN1; SMN2CYP1A2CYP3A4
SCHEMBL7722448 0.83 CYP4F2 (0.70) CYP4F2CYP4A11SMN1; SMN2CYP1A2CYP3A4
SCHEMBL4270902 0.81 CYP4F2 (0.64) CYP4F2CYP4A11SMN1; SMN2CYP1A2CYP3A4
SCHEMBL8851552 0.81 CYP4F2 (0.68) CYP4F2CYP4A11SMN1; SMN2CYP1A2CYP3A4
SCHEMBL11588447 0.81 CYP4F2 (0.68) CYP4F2CYP4A11SMN1; SMN2CYP1A2CYP3A4
SCHEMBL9157019 0.81 CYP4F2 (0.64) CYP4F2CYP4A11SMN1; SMN2CYP1A2CYP3A4
SCHEMBL1511092 0.81 CYP4F2 (0.64) CYP4F2CYP4A11SMN1; SMN2CYP1A2CYP3A4
SCHEMBL5132516 0.80 PKM (0.56) CYP4F2CYP4A11SMN1; SMN2CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5717094-A 6-THIOCHROMANYL-ETHYNE, 6-CHROMANYL ETHYNE AND 6-TETRAHYDROQUINOLINYL ETHYNE OR THEIR METAL SALTS ARE REACTED WITH SUITABLE HALO SUBSTITUTED PHENYL OR HETEROARYL COMPUNDS ALLERGAN (US) 1998-02-10 US disclosed
EP-0419132-B1 Process and intermediates for preparing compounds having a disubstituted acetylene moiety and retinoic acid-like biological activity ALLERGAN INC (US) 1995-09-06 EP disclosed
US-5248777-A Inhibitors of ornithine decarboxylase ALLERGAN, INC. (US) 1993-09-28 US disclosed
US-5053523-A Chemical intermediate for compounds having retinoic acid-like activity ALLERGAN, INC. (US) 1991-10-01 US disclosed
US-5023341-A Acetylene thiochroman ALLERGAN, INC. (US) 1991-06-11 US disclosed
EP-0419132-A2 Process and intermediates for preparing compounds having a disubstituted acetylene moiety and retinoic acid-like biological activity ALLERGAN, INC. (US) 1991-03-27 EP disclosed