SCHEMBL8564353

SCHEMBL8564353

Cc1ccc(S(=O)(=O)OC(=O)c2cn(C3CC3)c3c(Cl)c(N4CCC(N)C4)c(F)cc3c2=O)cc1

nearest known ligand 0.68

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.68
POLB P06746 2/20 0.68
OPRM1 P35372 2/20 0.68
CHRM2 P08172 1/20 0.68
CHRM1 P11229 1/20 0.68
OPRD1 P41143 1/20 0.68
KCNH2 Q12809 4/20 0.46
TOP1 P11387 4/20 0.43
TDP1 Q9NUW8 2/20 0.42
KDM4E B2RXH2 1/20 0.42
PRKD3 O94806 1/20 0.42
HPGD P15428 1/20 0.42
ALOX15 P16050 1/20 0.42
CLK2 P49760 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CLK4 Q9HAZ1 1/20 0.42
TOP2A P11388 6/20 0.41
TOP2B Q02880 4/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Clinafloxacin SCHEMBL8564349 0.88 ALDH1A1 (0.80) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL8128297 0.85 ALDH1A1 (0.64) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL16518620 0.83 ALDH1A1 (0.84) ALDH1A1POLBOPRM1CHRM2CHRM1
Clinafloxacin SCHEMBL28466331 0.82 ALDH1A1 (0.90) ALDH1A1POLBOPRM1CHRM2CHRM1
Clinafloxacin SCHEMBL8566142 0.82 ALDH1A1 (0.93) ALDH1A1POLBOPRM1CHRM2CHRM1
Clinafloxacin SCHEMBL33960 0.82 ALDH1A1 (1.00) ALDH1A1POLBOPRM1CHRM2CHRM1
Clinafloxacin SCHEMBL29360508 0.82 ALDH1A1 (1.00) ALDH1A1POLBOPRM1CHRM2CHRM1
Clinafloxacin SCHEMBL8596801 0.82 ALDH1A1 (1.00) ALDH1A1POLBOPRM1CHRM2CHRM1
Clinafloxacin SCHEMBL33959 0.82 ALDH1A1 (1.00) ALDH1A1POLBOPRM1CHRM2CHRM1
Clinafloxacin SCHEMBL5571098 0.81 ALDH1A1 (0.98) ALDH1A1POLBOPRM1CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5723627-A BACTERICIDES BAYER AKTIENGESELLSCHAFT (DE) 1998-03-03 US disclosed
US-5648493-A MULTISTAGE PROCESS BY CONDENSING AN OXO COMPOUND WITH AN AMINO COMPOUND TO PRODUCE AN IMINE THEN REACTING WITH AN OXO QUINOLINE CARBOXYLIC ACID BAYER AKTIENGESELLSCHAFT (DE) 1997-07-15 US disclosed
US-5061712-A BACTERICIDES BAYER AKTIENGESELLSCHAFT (DE) 1991-10-29 US disclosed