SCHEMBL856538

SCHEMBL856538

CCCc1c(C)nc(CN(C)C)nc1Cl

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.34
HTT P42858 1/20 0.30
KMT2A Q03164 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
TLR8 Q9NR97 1/20 0.30
TLR7 Q9NYK1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15434648 0.87 TLR8 (0.33) ALDH1A1HTTKMT2ASMN1; SMN2L3MBTL1
SCHEMBL855416 0.86 CYP1A2 (0.31)
SCHEMBL16461836 0.77 MAPT (0.31) HTTSMN1; SMN2L3MBTL1
SCHEMBL15429642 0.77
SCHEMBL855415 0.76
SCHEMBL857230 0.76 SLC6A2 (0.31)
SCHEMBL9289682 0.75 ALDH1A1 (0.31) ALDH1A1TLR8TLR7
SCHEMBL4980998 0.74 ALDH1A1 (0.39) ALDH1A1
SCHEMBL857121 0.74 PDK2 (0.43) ALDH1A1HTTKMT2ASMN1; SMN2L3MBTL1
SCHEMBL9287280 0.73 METAP2 (0.33) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2432779-A1 BENZOXAZEPINES BASED P13K/MT0R INHIBITORS AGAINST PROLIFERATIVE DISEASES Exelixis, Inc. (US) 2012-03-28 EP disclosed
WO-2010135524-A1 BENZOXAZEPINES BASED P13K/MT0R INHIBITORS AGAINST PROLIFERATIVE DISEASES EXELIXIS, INC. (US) 2010-11-25 WO disclosed