SCHEMBL8565866

SCHEMBL8565866

COc1nc2cc([N+](=O)[O-])cc(CC(CC(N)=O)C(N)=O)c2nc1OC

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
CYP3A4 P08684 1/20 0.33
MAPT P10636 5/20 0.32
PLA2G1B P04054 1/20 0.32
ATG4B Q9Y4P1 1/20 0.32
POLB P06746 2/20 0.32
HTT P42858 2/20 0.32
BACE1 P56817 1/20 0.32
ALDH1A1 P00352 3/20 0.32
KMT2A Q03164 3/20 0.32
MEN1 O00255 2/20 0.32
GAA P10253 1/20 0.32
PKM P14618 1/20 0.31
ALOX5 P09917 1/20 0.31
NPC1 O15118 1/20 0.31
LMNA P02545 1/20 0.31
AHR P35869 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8565855 0.93 POLB (0.33) CYP19A1SMN1; SMN2CYP3A4MAPTPOLB
SCHEMBL8568657 0.85 CYP3A4 (0.34) CYP19A1SMN1; SMN2CYP3A4MAPTPOLB
SCHEMBL5973535 0.78 POLB (0.41) CYP19A1MAPTPOLBHTTBACE1
SCHEMBL8078887 0.78 POLB (0.41) CYP19A1SMN1; SMN2MAPTPOLBHTT
SCHEMBL8086955 0.76 TRPV1 (0.37) SMN1; SMN2MAPTPOLBALDH1A1KMT2A
SCHEMBL8078889 0.76 HTT (0.39) CYP19A1SMN1; SMN2MAPTPOLBHTT
SCHEMBL5973317 0.75 NQO2 (0.40) CYP19A1MAPTPOLBHTTALDH1A1
SCHEMBL8090408 0.74 KMT2A (0.41) SMN1; SMN2MAPTALDH1A1KMT2AMEN1
SCHEMBL27462958 0.73 GRK6 (0.37) MAPTPOLBALDH1A1KMT2AMEN1
SCHEMBL27440732 0.73 NQO2 (0.38) CYP19A1SMN1; SMN2MAPTPOLBHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0853617-A1 NOVEL 2,3-DIOXO-1,2,3,4-TETRAHYDRO-QUINOYXALINYL DERIVATIVES Novartis AG (CH) 1998-07-22 EP disclosed
WO-1997008155-A1 NOVEL 2,3-DIOXO-1,2,3,4-TETRAHYDRO-QUINOYXALINYL DERIVATIVES NOVARTIS AG (CH) 1997-03-06 WO disclosed