SCHEMBL8568657

SCHEMBL8568657

COc1nc2cc([N+](=O)[O-])cc(CC(OC)C(N)=O)c2nc1OC

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CYP19A1 P11511 1/20 0.34
POLB P06746 2/20 0.33
HTT P42858 2/20 0.33
BACE1 P56817 1/20 0.33
MAPT P10636 4/20 0.32
KMT2A Q03164 2/20 0.32
PKM P14618 1/20 0.32
ALDH1A1 P00352 1/20 0.32
ALOX5 P09917 1/20 0.32
NPC1 O15118 1/20 0.32
LMNA P02545 1/20 0.32
MEN1 O00255 1/20 0.32
AHR P35869 1/20 0.32
SLC2A1 P11166 1/20 0.32
TDP1 Q9NUW8 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8565866 0.85 CYP19A1 (0.33) CYP3A4SMN1; SMN2CYP19A1POLBHTT
SCHEMBL8565855 0.84 POLB (0.33) CYP3A4SMN1; SMN2CYP19A1POLBHTT
SCHEMBL8078887 0.80 POLB (0.41) SMN1; SMN2CYP19A1POLBHTTMAPT
SCHEMBL5973535 0.80 POLB (0.41) CYP19A1POLBHTTBACE1MAPT
SCHEMBL8078889 0.77 HTT (0.39) SMN1; SMN2CYP19A1POLBHTTMAPT
SCHEMBL5973317 0.77 NQO2 (0.40) CYP19A1POLBHTTMAPTKMT2A
SCHEMBL8090408 0.76 KMT2A (0.41) SMN1; SMN2MAPTKMT2APKMALDH1A1
SCHEMBL8086955 0.75 TRPV1 (0.37) SMN1; SMN2POLBMAPTKMT2AALDH1A1
SCHEMBL27462958 0.75 GRK6 (0.37) POLBMAPTKMT2APKMALDH1A1
SCHEMBL27440732 0.75 NQO2 (0.38) SMN1; SMN2CYP19A1POLBHTTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0853617-A1 NOVEL 2,3-DIOXO-1,2,3,4-TETRAHYDRO-QUINOYXALINYL DERIVATIVES Novartis AG (CH) 1998-07-22 EP disclosed
WO-1997008155-A1 NOVEL 2,3-DIOXO-1,2,3,4-TETRAHYDRO-QUINOYXALINYL DERIVATIVES NOVARTIS AG (CH) 1997-03-06 WO disclosed