SCHEMBL8566080

SCHEMBL8566080

CCOc1cc2c(Nc3ccc(OC)cc3)c(Br)cnc2nc1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 2/20 0.43
PDE4D Q08499 1/20 0.43
DHFR P00374 1/20 0.42
MAP2K1 Q02750 1/20 0.40
STK4 Q13043 1/20 0.40
TP53 P04637 2/20 0.40
CSF1R P07333 1/20 0.39
MAPT P10636 3/20 0.39
KMT2A Q03164 3/20 0.39
MEN1 O00255 1/20 0.39
GAA P10253 1/20 0.39
TBK1 Q9UHD2 2/20 0.39
POLB P06746 3/20 0.39
RAD52 P43351 2/20 0.39
KDM4E B2RXH2 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
KDM1A O60341 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8564884 0.98 MAP2K1 (0.41) PDE4BPDE4DDHFRMAP2K1STK4
SCHEMBL8561356 0.89 PDE4B (0.44) PDE4BPDE4DDHFRMAP2K1STK4
Hydrochloric Acid SCHEMBL8561034 0.87 PDE4B (0.43) PDE4BPDE4DDHFRMAP2K1STK4
SCHEMBL8563461 0.85 PDE4B (0.41) PDE4BPDE4DDHFRMAP2K1STK4
SCHEMBL8325684 0.84 MAP2K1 (0.61) MAP2K1STK4EGFRERBB2
SCHEMBL8564146 0.83 CSF1R (0.50) PDE4BSTK4CSF1RMAPTKMT2A
SCHEMBL9542093 0.83 PDE4B (0.47) PDE4BTP53MAPTKMT2AMEN1
SCHEMBL8563378 0.83 PDE4B (0.59) PDE4BTP53CSF1RMAPTKMT2A
SCHEMBL8565303 0.83 CSF1R (0.62) PDE4BCSF1REGFRERBB2
SCHEMBL8559603 0.83 DHFR (0.41) PDE4BPDE4DDHFRMAP2K1STK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618916-B1 ANTI-RHEUMATIC NAPHTHYRIDINE DERIVATIVES KNOLL AG (DE) 1998-09-23 EP disclosed
US-5464781-A TREATING RHEUMATIC DISEASES THE BOOTS COMPANY PLC (GB) 1995-11-07 US disclosed