SCHEMBL8566878

SCHEMBL8566878

O=C1Cc2cc(Cl)ccc2C(=O)N1Cc1ccccc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 7/20 0.71
MEN1 O00255 6/20 0.71
CASP6 P55212 2/20 0.71
APAF1 O14727 3/20 0.71
ALDH1A1 P00352 3/20 0.71
MAPT P10636 3/20 0.71
HPGD P15428 2/20 0.71
GAA P10253 2/20 0.53
CASP3 P42574 2/20 0.53
SENP8 Q96LD8 1/20 0.53
SENP7 Q9BQF6 1/20 0.53
SENP6 Q9GZR1 1/20 0.53
BLM P54132 2/20 0.52
CASP1 P29466 1/20 0.52
RAB9A P51151 1/20 0.52
CASP7 P55210 1/20 0.52
HSD17B10 Q99714 1/20 0.52
ALDH2 P05091 1/20 0.52
ALDH3A1 P30838 1/20 0.52
MDH2 P40926 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29609544 0.83 KMT2A (1.00) KMT2AMEN1CASP6APAF1ALDH1A1
SCHEMBL2586644 0.83 KMT2A (1.00) KMT2AMEN1CASP6APAF1ALDH1A1
SCHEMBL8207403 0.80 KMT2A (0.63) KMT2AMEN1CASP6APAF1ALDH1A1
SCHEMBL28350022 0.79 KMT2A (0.65) KMT2AMEN1ALDH1A1MAPTHPGD
SCHEMBL30378020 0.79 KMT2A (0.65) KMT2AMEN1ALDH1A1MAPTHPGD
SCHEMBL2023150 0.77 GRM5 (0.50) KMT2AMEN1CASP6APAF1ALDH1A1
SCHEMBL1260656 0.75 KMT2A (0.45) KMT2AMEN1CASP6APAF1ALDH1A1
SCHEMBL9918982 0.72 SRD5A1 (0.50) KMT2AMEN1CASP6GAA
SCHEMBL5807332 0.72 KMT2A (0.59) KMT2AMEN1CASP6APAF1ALDH1A1
SCHEMBL29648466 0.72 ALDH1A1 (0.78) CASP6APAF1ALDH1A1MAPTCASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5741798-A 2-benzyl-4-sulfonyl-4H-isoquinolin-1,3-diones and their use as antiinflammatory agents BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 1998-04-21 US disclosed
WO-1997046532-A1 2-BENZYL-4-SULFONYL-4H-ISOQUINOLIN-1,3-DIONES AND THEIR USE AS ANTI-INFLAMMATORY AGENTS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 1997-12-11 WO disclosed