SCHEMBL8567007

SCHEMBL8567007

CCC(Cn1ccc2nc(N)nc(N)c21)c1ccc(C(=O)N[C@H](CCC(=O)O)C(=O)O)o1

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DHFR P00374 8/20 0.47
ATIC P31939 4/20 0.45
SHMT1 P34896 4/20 0.45
SHMT2 P34897 4/20 0.45
GART P22102 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8567001 1.00 DHFR (0.47) DHFRATICSHMT1SHMT2GART
SCHEMBL8562553 0.93 ATIC (0.48) DHFRATICSHMT1SHMT2GART
SCHEMBL8562562 0.93 ATIC (0.48) DHFRATICSHMT1SHMT2GART
SCHEMBL8571458 0.90 DHFR (0.48) DHFRATICSHMT1SHMT2GART
SCHEMBL8571474 0.90 DHFR (0.48) DHFRATICSHMT1SHMT2GART
SCHEMBL9001772 0.86 ATIC (0.63) DHFRATICSHMT1SHMT2GART
SCHEMBL8571094 0.86 ATIC (0.49) DHFRATICSHMT1SHMT2GART
SCHEMBL8571085 0.86 ATIC (0.49) DHFRATICSHMT1SHMT2GART
SCHEMBL8564196 0.85 DHFR (0.58) DHFRATICSHMT1SHMT2GART
SCHEMBL8564205 0.85 DHFR (0.58) DHFRATICSHMT1SHMT2GART

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530579-B1 Condensed pyrimidine derivatives antitumor agents EISAI CO LTD (JP) 1998-11-11 EP disclosed
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed