SCHEMBL8567170

SCHEMBL8567170

N#Cc1ccc2c(c1)CCC(N1CCC3(CC1)CC(=O)c1cc([N+](=O)[O-])c(N)cc1O3)C2

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.47
CYP11B2 P19099 1/20 0.39
CA1 P00915 12/20 0.38
CA2 P00918 12/20 0.38
CA7 P43166 12/20 0.38
CA9 Q16790 12/20 0.38
HTR2A P28223 2/20 0.37
KCNJ1 P48048 1/20 0.37
DRD2 P14416 1/20 0.37
EPHX1 P07099 1/20 0.36
EPHX2 P34913 1/20 0.36
SCN5A Q14524 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8569179 0.90 KCNH2 (0.52) KCNH2CYP11B2HTR2AKCNJ1DRD2
SCHEMBL8565862 0.88 DRD2 (0.48) CA1CA2CA7CA9HTR2A
SCHEMBL8570143 0.83 CA1 (0.45) CA1CA2CA7CA9HTR2A
SCHEMBL8567782 0.83 KCNH2 (0.50) KCNH2CYP11B2HTR2AKCNJ1DRD2
Hydrochloric Acid SCHEMBL8571057 0.82 CA1 (0.48) CA1CA2CA7CA9HTR2A
Hydrochloric Acid SCHEMBL8564675 0.82 KCNH2 (0.49) KCNH2CYP11B2HTR2AKCNJ1DRD2
SCHEMBL8563772 0.80 KCNH2 (0.58) KCNH2CYP11B2CA1CA2CA7
SCHEMBL8804765 0.79 KCNH2 (0.53) KCNH2CYP11B2CA1CA2CA7
SCHEMBL8566094 0.79 KCNH2 (0.48) KCNH2CYP11B2HTR2AKCNJ1DRD2
Hydrochloric Acid SCHEMBL8806196 0.78 KCNH2 (0.52) KCNH2CYP11B2CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431943-B1 Spiro(pyran)piperidine derivatives MERCK & CO INC (US) 1998-07-15 EP disclosed
US-5633247-A ANTIARRTHYMIA AGENT MERCK & CO., INC. (US) 1997-05-27 US disclosed
US-5206240-A Antiarrhythmia agents MERCK & CO., INC. (US) 1993-04-27 US disclosed