SCHEMBL8567192

SCHEMBL8567192

COC(=O)CCC1CNC(=O)N(c2ccc3c(c2)CCN(C(=O)C(F)(F)F)CC3)C1C1CCCCC1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.37
ESR2 Q92731 3/20 0.37
HDAC6 Q9UBN7 4/20 0.33
FHIT P49789 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4D Q08499 1/20 0.32
CCR2 P41597 6/20 0.31
CCR1 P32246 5/20 0.31
P2RX3 P56373 1/20 0.31
CYP2D6 P10635 1/20 0.30
TMEM97 Q5BJF2 1/20 0.30
SIGMAR1 Q99720 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8558842 0.85 HTR6 (0.33) FHITCCR2CCR1P2RX3CYP2D6
SCHEMBL8563251 0.78 ESR1 (0.39) ESR1ESR2HDAC6FHITPDE4B
SCHEMBL8559448 0.78 ESR1 (0.39) ESR1ESR2HDAC6PDE4BPDE4D
SCHEMBL8567196 0.78 ESR1 (0.39) ESR1ESR2HDAC6FHITPDE4B
SCHEMBL8561833 0.75 ESR1 (0.39) ESR1ESR2HDAC6
SCHEMBL8559207 0.74 MAPT (0.43) ESR1ESR2CYP2D6
SCHEMBL8563245 0.74 ESR1 (0.38) ESR1ESR2HDAC6PDE4BPDE4D
SCHEMBL8564189 0.72 ESR1 (0.41) ESR1ESR2HDAC6PDE4BPDE4D
SCHEMBL8564198 0.72 ESR1 (0.41) ESR1ESR2HDAC6PDE4BPDE4D
SCHEMBL8559199 0.72 ESR1 (0.39) ESR1ESR2PDE4BPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5827849-A HAVING INHIBITORY EFFECT ON INFLAMMATION AND BONE DEGRADATION, ANTITHROMBOTIC, ANTIAGGREGATORY AND TUMOR- OR METASTASIS-INHIBITING EFFECT KARL THOMAE GMBH (DE) 1998-10-27 US disclosed