SCHEMBL8567463

SCHEMBL8567463

NCC(=O)N(CC(=O)O)C(=O)C1CCCN1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SCN4A P35499 1/20 0.37
NOS2 P35228 2/20 0.36
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36
PRCP P42785 1/20 0.33
DPP4 P27487 6/20 0.32
GLI1 P08151 2/20 0.32
DPP8 Q6V1X1 4/20 0.31
DPP9 Q86TI2 4/20 0.31
MEN1 O00255 1/20 0.31
BLM P54132 1/20 0.31
KMT2A Q03164 1/20 0.31
FAP Q12884 1/20 0.31
DPP7 Q9UHL4 1/20 0.31
ARG1 P05089 1/20 0.30
ARG2 P78540 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6156985 0.88 NOS2 (0.40) SCN4ANOS2NOS3NOS1PRCP
SCHEMBL3359438 0.87 SCN4A (0.42) SCN4ANOS2NOS3NOS1PRCP
SCHEMBL16620345 0.79 SCN4A (0.38) SCN4ANOS2NOS3NOS1PRCP
SCHEMBL194737 0.78 SCN4A (0.43) SCN4A
SCHEMBL27740316 0.76 SCN4A (0.33) SCN4ANOS2NOS3NOS1
SCHEMBL28367481 0.76 SCN4A (0.41) SCN4ANOS2NOS3NOS1PRCP
SCHEMBL10793329 0.75 GSR (0.38) SCN4ADPP4DPP8DPP9FAP
SCHEMBL30851509 0.75 NOS2 (0.39) SCN4ANOS2NOS3NOS1PRCP
SCHEMBL8788154 0.74 SCN4A (0.47) SCN4ANOS2NOS3NOS1PRCP
SCHEMBL29772688 0.74 SCN4A (0.47) SCN4ANOS2NOS3NOS1PRCP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0142231-B1 PROCESS FOR PRODUCING SEQUENTIAL POLYAMINO ACID RESIN NITTO BOSEKI CO., LTD. (JP) 1987-11-11 EP claimed
EP-0142231-A1 Process for producing sequential polyamino acid resin NITTO BOSEKI CO., LTD. (JP) 1985-05-22 EP claimed
EP-0545991-B1 PEPTIDES THAT BLOCK HUMAN IMMUNODEFICIENCY VIRUS INFECTIONS AND METHODS OF USE THEREOF VAHLNE ANDERS (SE) 1998-12-02 EP disclosed
US-5627035-A Peptides that block human immunodeficiency virus and methods of use thereof SYNTELLO VACCINE DEVELOPMENT AB (SE) 1997-05-06 US disclosed
EP-0545991-A1 PEPTIDES THAT BLOCK HUMAN IMMUNODEFICIENCY VIRUS INFECTIONS AND METHODS OF USE THEREOF VAHLNE, Anders (SE) 1993-06-16 EP disclosed
WO-1992003147-A1 PEPTIDES THAT BLOCK HUMAN IMMUNODEFICIENCY VIRUS INFECTIONS AND METHODS OF USE THEREOF SYNTELLO VACCIN DEVELOPMENT KB (SE) 1992-03-05 WO disclosed