SCHEMBL8568262

SCHEMBL8568262

CNC(=O)c1cccnc1Oc1ccccc1

nearest known ligand 0.74

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.74
TDP1 Q9NUW8 1/20 0.71
MAPK8 P45983 4/20 0.71
KMT2A Q03164 1/20 0.64
GAA P10253 3/20 0.62
MAPT P10636 1/20 0.62
KDM4E B2RXH2 1/20 0.58
POLB P06746 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5094162 0.87 ALDH1A1 (0.60) ALDH1A1TDP1MAPK8KMT2AGAA
SCHEMBL5213184 0.85 ALDH1A1 (1.00) ALDH1A1TDP1MAPK8KMT2AGAA
SCHEMBL4558530 0.84 ALDH1A1 (0.68) ALDH1A1TDP1MAPK8KMT2AGAA
SCHEMBL4939060 0.84 KMT2A (0.82) ALDH1A1TDP1MAPK8KMT2AGAA
SCHEMBL2488732 0.83
SCHEMBL20818012 0.83 TDP1 (1.00) ALDH1A1TDP1MAPK8KMT2AGAA
SCHEMBL7310026 0.83 MAPK8 (1.00) ALDH1A1TDP1MAPK8GAA
SCHEMBL13692388 0.83 TDP1 (0.72) ALDH1A1TDP1MAPK8KMT2AGAA
SCHEMBL861902 0.82 TDP1 (0.71) ALDH1A1TDP1MAPK8KMT2AGAA
SCHEMBL5216347 0.81 ALDH1A1 (0.68) ALDH1A1TDP1MAPK8KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5846990-A Substituted biphenyl isoxazole sulfonamides BRISTOL-MYERS SQUIBB CO. (US) 1998-12-08 US disclosed