SCHEMBL7310026

SCHEMBL7310026

O=C(NCc1ccccc1)c1cccnc1Oc1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 3/20 1.00
ALDH1A1 P00352 1/20 0.71
TDP1 Q9NUW8 1/20 0.60
GAA P10253 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14193488 0.90 MAPK8 (0.82) MAPK8
SCHEMBL7319190 0.88 MAPK8 (0.78) MAPK8ALDH1A1
SCHEMBL7307728 0.88 MAPK8 (0.78) MAPK8ALDH1A1
SCHEMBL8756555 0.88 MAPK8 (0.78) MAPK8ALDH1A1
SCHEMBL10073050 0.87 MAPK8 (0.77) MAPK8ALDH1A1
SCHEMBL2485262 0.86 MAPK8 (0.75) MAPK8
SCHEMBL7317640 0.86 MAPK8 (0.75) MAPK8
SCHEMBL7366565 0.85 MAPK8 (0.73) MAPK8ALDH1A1
SCHEMBL7168843 0.84 MAPK8 (0.72) MAPK8GAA
SCHEMBL8568262 0.83 ALDH1A1 (0.74) MAPK8ALDH1A1TDP1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0357316-B1 ANTIDEPRESSANT N-SUBSTITUTED NICOTINAMIDE COMPOUNDS PFIZER INC. (US) 1993-04-14 EP disclosed
EP-0357316-A1 Antidepressant N-substituted nicotinamide compounds PFIZER INC. (US) 1990-03-07 EP disclosed
US-4861891-A Antidepressant N-substituted nicotinamide compounds PFIZER INC. (US) 1989-08-29 US disclosed