SCHEMBL8569042

SCHEMBL8569042

CC(Cn1ccc2nc(N)nc(N)c21)c1ccc(C(=O)N[C@H](CCC(=O)O)C(=O)O)s1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ATIC P31939 9/20 0.51
SHMT1 P34896 9/20 0.51
SHMT2 P34897 9/20 0.51
GART P22102 7/20 0.50
DHFR P00374 6/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8569034 1.00 ATIC (0.51) ATICSHMT1SHMT2GARTDHFR
SCHEMBL8570075 0.92 ATIC (0.54) ATICSHMT1SHMT2GARTDHFR
SCHEMBL8570081 0.92 ATIC (0.54) ATICSHMT1SHMT2GARTDHFR
SCHEMBL8570677 0.90 ATIC (0.49) ATICSHMT1SHMT2GARTDHFR
SCHEMBL8570681 0.90 ATIC (0.49) ATICSHMT1SHMT2GARTDHFR
SCHEMBL9001763 0.86 ATIC (0.69) ATICSHMT1SHMT2GARTDHFR
SCHEMBL8571212 0.86 ATIC (0.53) ATICSHMT1SHMT2GARTDHFR
SCHEMBL8571222 0.86 ATIC (0.53) ATICSHMT1SHMT2GARTDHFR
SCHEMBL8571414 0.84 DHFR (0.57) ATICSHMT1SHMT2GARTDHFR
SCHEMBL8571420 0.84 DHFR (0.57) ATICSHMT1SHMT2GARTDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530579-B1 Condensed pyrimidine derivatives antitumor agents EISAI CO LTD (JP) 1998-11-11 EP disclosed
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed