SCHEMBL8569847

SCHEMBL8569847

COC(=O)c1ccc(OC)c(NCC(=N)c2ccc(OC)cc2)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.57
KMT2A Q03164 3/20 0.54
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
GAA P10253 2/20 0.49
TP53 P04637 1/20 0.49
HDAC8 Q9BY41 2/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
MEN1 O00255 2/20 0.47
NPC1 O15118 1/20 0.47
MAPT P10636 3/20 0.46
POLB P06746 2/20 0.46
ALDH1A1 P00352 5/20 0.46
TSHR P16473 2/20 0.45
NPSR1 Q6W5P4 1/20 0.45
KDM4E B2RXH2 1/20 0.45
HPGD P15428 1/20 0.45
MDH1 P40925 1/20 0.45
MDH2 P40926 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8571489 0.90 HDAC8 (0.51) CYP2C9KMT2AGAAHDAC8HDAC1
SCHEMBL8574648 0.89 ALDH1A1 (0.45) CYP2C9KMT2AGAAHDAC8HDAC1
SCHEMBL7367017 0.88 KMT2A (0.55) CYP2C9KMT2ACA1CA2GAA
SCHEMBL7363238 0.84 MAPT (0.50) CYP2C9KMT2AHDAC8HDAC1HDAC6
SCHEMBL7366511 0.82 ALDH1A1 (0.53) CYP2C9KMT2AGAAHDAC8HDAC1
SCHEMBL7364156 0.79 ALDH1A1 (0.50) CYP2C9KMT2AGAAHDAC8HDAC1
SCHEMBL7359031 0.78 MAPT (0.47) CYP2C9KMT2AGAAHDAC8HDAC1
SCHEMBL1553492 0.78 MDH1 (0.59) CYP2C9KMT2ACA1CA2GAA
SCHEMBL1553048 0.78 KMT2A (0.55) CYP2C9KMT2ACA1CA2GAA
SCHEMBL8569761 0.78 HDAC8 (0.53) CYP2C9KMT2AGAAHDAC8HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998005327-A1 SUBSTITUTED AROMATIC COMPOUNDS RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1998-02-12 WO disclosed