SCHEMBL8570715

SCHEMBL8570715

CCOC(=O)CCc1ccc(C(=O)OC(C)(C)C)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 2/20 0.60
CYP4A11 Q02928 2/20 0.60
CYP4Z1 Q86W10 1/20 0.49
EPHX2 P34913 1/20 0.48
LMNA P02545 4/20 0.45
MAPT P10636 3/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
NAMPT P43490 1/20 0.43
TDP1 Q9NUW8 3/20 0.43
MAPK1 P28482 2/20 0.43
GAA P10253 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43
CA12 O43570 2/20 0.42
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA9 Q16790 2/20 0.42
CA14 Q9ULX7 2/20 0.42
ESR1 P03372 1/20 0.42
CA7 P43166 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7662083 0.89 CYP4A11 (0.48) CYP4F2CYP4A11CYP4Z1EPHX2LMNA
SCHEMBL7766764 0.86 CYP4F2 (0.70) CYP4F2CYP4A11CYP4Z1EPHX2LMNA
SCHEMBL31635260 0.85 LMNA (0.56) CYP4F2CYP4A11CYP4Z1LMNAMAPT
SCHEMBL7582610 0.85 ADRB2 (0.48) CYP4F2CYP4A11LMNAMAPTL3MBTL1
SCHEMBL16838984 0.82 SMN1; SMN2 (0.52) CYP4F2CYP4A11LMNAMAPTL3MBTL1
SCHEMBL68902 0.82 CYP4F2 (0.85) CYP4F2CYP4A11CYP4Z1EPHX2LMNA
SCHEMBL3790673 0.81 NR1H4 (0.51) EPHX2LMNAL3MBTL1NPSR1CA12
SCHEMBL13891334 0.81 PLK1 (0.51) CYP4F2CYP4A11MAPTL3MBTL1GAA
SCHEMBL18608207 0.81 CA1 (0.63) LMNAMAPTTDP1MAPK1NPSR1
SCHEMBL879130 0.81 CYP4F2 (0.77) CYP4F2CYP4A11CYP4Z1EPHX2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530579-B1 Condensed pyrimidine derivatives antitumor agents EISAI CO LTD (JP) 1998-11-11 EP disclosed
US-5688800-A ANTITUMOR AGENTS EISAI CO., LTD. (JP) 1997-11-18 US disclosed
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed
US-4742052-A Antibacterial β-lactam compounds SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1988-05-03 US disclosed
EP-0070204-A2 Carboxylic beta-lactam compounds and the preparation thereof SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1983-01-19 EP disclosed