SCHEMBL8570827

SCHEMBL8570827

CON(C)C(=O)c1cc(Cl)ccc1OCc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 7/20 0.56
APP P05067 1/20 0.52
NPC1 O15118 1/20 0.52
ALDH1A1 P00352 1/20 0.52
MAPT P10636 1/20 0.52
HPGD P15428 1/20 0.52
HTT P42858 1/20 0.52
RAB9A P51151 1/20 0.52
MDM2 Q00987 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
GPR55 Q9Y2T6 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
KMT2A Q03164 1/20 0.52
LRRK2 Q5S007 2/20 0.51
TSHR P16473 1/20 0.50
CYP2C9 P11712 2/20 0.48
MRGPRX4 Q96LA9 2/20 0.47
KCNA3 P22001 1/20 0.47
AKR1C3 P42330 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4480514 0.85 APP (0.52) APPNPC1ALDH1A1MAPTHPGD
SCHEMBL31055984 0.85 APP (0.52) PTGER1APPNPC1HPGDRAB9A
SCHEMBL2290346 0.84 TRPM8 (0.55) PTGER1APPNPC1HTTKMT2A
SCHEMBL31056340 0.83 APP (0.58) APPNPC1ALDH1A1HPGDHTT
SCHEMBL8571163 0.83 TSHR (0.49) NPC1ALDH1A1MAPTHPGDHTT
SCHEMBL9789583 0.82 PTGER1 (0.61) PTGER1HPGDKMT2ALRRK2CYP2C9
SCHEMBL4722050 0.81 PTGER1 (0.64) PTGER1MAPTSMN1; SMN2L3MBTL1KMT2A
SCHEMBL29836110 0.81 PTGER1 (0.64) PTGER1MAPTSMN1; SMN2L3MBTL1KMT2A
SCHEMBL487486 0.81 PTGER1 (0.75) PTGER1ALDH1A1L3MBTL1KMT2ALRRK2
SCHEMBL2114834 0.81 PTGER1 (0.53) PTGER1APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739336-A SELECTIVE 5-HYDROXYTRYPTAMINE-2C RECEPTOR ANTAGONISTS SYNTEX (U.S.A.) INC. (US) 1998-04-14 US disclosed
WO-1997000872-A1 1,3,8-TRIAZA- AND 3,8-DIAZA-1-OXASPIRO(4,5)DECANE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 1997-01-09 WO disclosed