SCHEMBL8571007

SCHEMBL8571007

CC(C)(C)OC(=O)N1CCN(Cc2ccccc2)CC1COCc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.49
NR1H2 P55055 2/20 0.46
NR1H3 Q13133 2/20 0.46
AGTR2 P50052 1/20 0.44
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
CA4 P22748 2/20 0.41
CA9 Q16790 2/20 0.41
OPRD1 P41143 1/20 0.41
OPRK1 P41145 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
MAPK1 P28482 1/20 0.41
KLK7 P49862 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8571009 1.00 PARP1 (0.49) PARP1NR1H2NR1H3AGTR2CA1
SCHEMBL8238395 0.88 NR1H2 (0.43) PARP1NR1H2NR1H3AGTR2CA1
SCHEMBL28549464 0.87 PARP1 (0.46) PARP1NR1H2NR1H3AGTR2OPRD1
SCHEMBL12780700 0.86 SIGMAR1 (0.52) PARP1NR1H2NR1H3AGTR2CA1
SCHEMBL8448438 0.86 NR1H2 (0.58) PARP1NR1H2NR1H3AGTR2CA1
SCHEMBL8240100 0.86 SIGMAR1 (0.52) PARP1NR1H2NR1H3AGTR2CA1
SCHEMBL6975745 0.86 NR1H2 (0.48) PARP1NR1H2NR1H3AGTR2CA1
SCHEMBL6099695 0.86 NR1H2 (0.58) PARP1NR1H2NR1H3AGTR2CA1
SCHEMBL6975743 0.86 NR1H2 (0.48) PARP1NR1H2NR1H3AGTR2CA1
SCHEMBL26915001 0.85 NR1H2 (0.48) PARP1NR1H2NR1H3AGTR2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5736539-A ANITCARCINOGENIC AGENTS MERCK & CO., INC. (US) 1998-04-07 US disclosed
WO-1995000497-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 1995-01-05 WO disclosed