SCHEMBL8574241

SCHEMBL8574241

CCOC(CN(C(=O)Nc1ccc(CC(NC(=O)OC(C)(C)C)C(=O)OC)cc1)c1ccc(C#N)cc1)OCC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 7/20 0.41
CTSK P43235 6/20 0.41
NLRP3 Q96P20 1/20 0.41
CTSB P07858 2/20 0.40
CTSL P07711 1/20 0.40
KLK5 Q9Y337 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
CTSG P08311 1/20 0.38
CMA1 P23946 1/20 0.38
ITGB3 P05106 1/20 0.38
ITGB1 P05556 1/20 0.38
ITGAV P06756 1/20 0.38
ITGA2B P08514 1/20 0.38
ITGB5 P18084 1/20 0.38
PTPN1 P18031 1/20 0.38
PPARG P37231 1/20 0.38
PPARA Q07869 1/20 0.38
PSEN1 P49768 2/20 0.36
PSEN2 P49810 2/20 0.36
APH1B Q8WW43 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18920552 0.81 CTSS (0.58) CTSSCTSKNLRP3CTSBCTSL
SCHEMBL16935712 0.81 CTSS (0.58) CTSSCTSKNLRP3CTSBCTSL
SCHEMBL2617261 0.81 CTSS (0.58) CTSSCTSKNLRP3CTSBCTSL
SCHEMBL8910751 0.78 PSMB5 (0.44)
SCHEMBL539374 0.78 CTSS (0.62) CTSSCTSKNLRP3CTSBCTSL
SCHEMBL539373 0.78 CTSS (0.62) CTSSCTSKNLRP3CTSBCTSL
SCHEMBL8572808 0.78 RORC (0.43)
SCHEMBL23419674 0.77 CTSS (0.56) CTSSCTSKCTSBCTSLCTSG
SCHEMBL5151368 0.77 CTSS (0.56) CTSSCTSKCTSBCTSLCTSG
SCHEMBL31524193 0.76 CTSS (0.59) CTSSCTSKNLRP3CTSBCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5852192-A Cyclic urea derivatives, pharmaceutical compositions containing these compounds and processes for preparing them DR. KARL THOMAE GMBH (DE) 1998-12-22 US disclosed
US-5650424-A ANTIAGGLOMERANTS USING IMIDAZOLIDINDIONES DR. KARL THOMAE GMBH (DE) 1997-07-22 US disclosed
US-5478942-A Antiinflammatory agents, antiagglomerants KARL THOMAE GMBH (DE) 1995-12-26 US disclosed
US-5276049-A Treatment of thrombosis DR. KARL THOMAE GMBH (DE) 1994-01-04 US disclosed