SCHEMBL8574265

SCHEMBL8574265

COCCC(c1ccccc1)c1nc2c(OC)ccc(CC(=O)O)c2[nH]1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.37
TAS1R1 Q7RTX1 1/20 0.37
STING1 Q86WV6 1/20 0.36
HSD17B10 Q99714 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.35
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
HPGD P15428 2/20 0.34
ROCK2 O75116 4/20 0.34
ROCK1 Q13464 4/20 0.34
ADORA2A P29274 2/20 0.34
CNR2 P34972 2/20 0.34
MAOB P27338 1/20 0.34
KEAP1 Q14145 1/20 0.34
NFE2L2 Q16236 1/20 0.34
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8570001 0.91 HSD17B10 (0.36) STING1HSD17B10PTGDR2MEN1KMT2A
SCHEMBL1553351 0.85 PDE4A (0.38) TAS1R3TAS1R1MEN1KMT2AHPGD
SCHEMBL8574183 0.85 HSD17B10 (0.39) STING1HSD17B10PTGDR2MEN1KMT2A
SCHEMBL8574177 0.83 PDE4A (0.39) TAS1R3TAS1R1HPGDROCK2ROCK1
SCHEMBL1553472 0.83 PDE4A (0.39) TAS1R3TAS1R1HSD17B10HPGDROCK2
SCHEMBL8571923 0.81 PDE4A (0.45) STING1HSD17B10HPGDPDE4APDE4B
SCHEMBL8572847 0.78 PTGDR2 (0.41) PTGDR2MEN1KMT2ALMNA
SCHEMBL8569838 0.77 HSD17B10 (0.37) STING1HSD17B10PTGDR2MEN1KMT2A
SCHEMBL1553694 0.76 PDE4D (0.61) PDE4APDE4BPDE4CPDE4D
SCHEMBL1553052 0.76 PDE4D (0.61) PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998005327-A1 SUBSTITUTED AROMATIC COMPOUNDS RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1998-02-12 WO disclosed