SCHEMBL8574353

SCHEMBL8574353

Nc1nc2ccccc2cc1-c1ccccc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.74
NPC1 O15118 3/20 0.74
RAB9A P51151 3/20 0.74
MEN1 O00255 2/20 0.74
FGFR1 P11362 1/20 0.62
SRC P12931 1/20 0.62
ATM Q13315 1/20 0.57
ALDH1A1 P00352 6/20 0.51
KDM4E B2RXH2 5/20 0.51
TDP1 Q9NUW8 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
GAA P10253 3/20 0.50
TLR8 Q9NR97 3/20 0.50
SMARCA2 P51531 1/20 0.50
SMARCA4 P51532 1/20 0.50
PBRM1 Q86U86 1/20 0.50
IKBKB O14920 1/20 0.49
HPGD P15428 3/20 0.48
GLA P06280 2/20 0.48
LMNA P02545 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1767756 0.85 MEN1 (1.00) KMT2ANPC1RAB9AMEN1FGFR1
SCHEMBL22509831 0.85 KMT2A (0.71) KMT2ANPC1RAB9AMEN1FGFR1
SCHEMBL27590143 0.85 KMT2A (0.56) KMT2ANPC1RAB9AMEN1FGFR1
SCHEMBL807074 0.83 FGFR1 (0.57) KMT2ANPC1RAB9AMEN1FGFR1
SCHEMBL22509832 0.83 MEN1 (0.58) KMT2ANPC1RAB9AMEN1FGFR1
Hydrochloric Acid SCHEMBL789680 0.82 FGFR1 (0.55) KMT2ANPC1RAB9AMEN1FGFR1
SCHEMBL28156921 0.80 FGFR1 (0.62) KMT2ANPC1RAB9AMEN1FGFR1
SCHEMBL790060 0.80 FGFR1 (0.54) KMT2ANPC1RAB9AMEN1FGFR1
SCHEMBL28280373 0.78 FGFR1 (0.55) KMT2ANPC1RAB9AMEN1FGFR1
SCHEMBL29374375 0.78 PSMB5 (0.65) KMT2ANPC1RAB9AMEN1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101171009-A Treatment of parkinson's disease obstructive sleep apnea, dementia with lewy bodies, vascular dementia with non-imidazole alkylamines histamine h3- receptor ligands BIOPROJET SOC CIV (FR) 2008-04-30 CN claimed
US-11988661-B2 Rapid quantitative test to diagnose polycystic kidney disease UMC UTRECHT HOLDING, B.V. (NL) 2024-05-21 US disclosed
US-20210333266-A1 RAPID QUANTITATIVE ASSAY TO MEASURE CFTR FUNCTION IN A PRIMARY INTESTINAL CULTURE MODEL UMC UTRECHT HOLDING, B.V. (NL) 2021-10-28 US disclosed
US-11035852-B2 Identifying drug candidates for treating polycystic kidney disease using organoids generated from primary cells UMC UTRECHT HOLDING, B.V. (NL) 2021-06-15 US disclosed
CN-102812045-B Materials and methods for treating or preventing human epidermal growth factor receptor-3 (HER-3) related diseases 第三共欧洲有限公司 2018-04-13 CN disclosed
CN-103772373-B As the quinazoline analogs of receptor tyrosine kinase inhibitors 阿雷生物药品公司 2017-06-09 CN disclosed
CN-106432206-A Method for synthesizing lapatinib or intermediate 5-(4-hydroxy quinazoline)-furan-2-formaldehyde of lapatinib 成都美睿科生物科技有限公司 2017-02-22 CN disclosed
CN-106432205-A Method for synthesizing lapatinib or intermediate thereof 成都美睿科生物科技有限公司 2017-02-22 CN disclosed
CN-103228632-B Compounds as modulators of mutant CFTR proteins and their use in treating diseases associated with CFTR protein malfunction 波兰科学院生物化学与生物物理研究所 2016-08-31 CN disclosed
CN-104496840-A Compounds As Modulators Of A Mutant Cftr Protein And Their Use For Treating Diseases Associated With Cftr Protein Malfunction INST BIOCHEMII I BIOFIZYKI PAN 2015-04-08 CN disclosed
US-20140203270-A1 ORGANIC ELECTROLUMINESCENT ELEMENT MATERIAL HAVING SILICON-CONTAINING FOUR MEMBERED RING STRUCTURE, AND ORGANIC ELECTROLUMINESCENT ELEMENT NIPPON STEEL & SUMIKIN CHEMICAL CO., LTD. (JP) 2014-07-24 US disclosed
WO-2013130660-A1 AMIDES AS PIM INHIBITORS AMGEN INC. (US) 2013-09-06 WO disclosed
CN-103228632-A Compounds as modulators of mutant CFTR proteins and their use in treating diseases associated with CFTR protein malfunction INST BIOCHEMII I BIOFIZYKI PAN 2013-07-31 CN disclosed
CN-101171009-B Use of non-imidazole alkylamines histamine h3- receptor ligands in treatment of parkinson's disease obstructive sleep apnea, dementia with lewy bodies, vascular dementia BIOPROJET SOC CIV 2012-11-07 CN disclosed
US-8288410-B2 3-substituted quinolinium and 7H-indolo[2,3-c]quinolinium salts as new antiinfectives FLORIDA AGRICULTURAL AND MECHANICAL UNIVERSITY (US) 2012-10-16 US disclosed
US-20120165369-A1 3-SUBSTITUTED QUINOLINIUM AND 7H-INDOLO[2,3-c]QUINOLINIUM SALTS AS NEW ANTIINFECTIVES FLORIDA AGRICULTURAL AND MECHANICAL UNIVERSITY 2012-06-28 US disclosed
CN-101605543-A Compounds having activity in correcting mutant-CFTR processing and uses thereof UNIV CALIFORNIA (US) 2009-12-16 CN disclosed
CN-101605543-A Compounds having activity in correcting mutant-CFTR processing and uses thereof UNIV CALIFORNIA (US) 2009-12-16 CN disclosed
CN-101171009-A Treatment of parkinson's disease obstructive sleep apnea, dementia with lewy bodies, vascular dementia with non-imidazole alkylamines histamine h3- receptor ligands BIOPROJET SOC CIV (FR) 2008-04-30 CN disclosed
WO-1998000750-A1 PROCESS FOR PRODUCING LIQUID CRYSTAL ALIGNMENT LAYER AND LIQUID CRYSTAL DISPLAY DEVICE WITH THE USE OF THE SAME HOECHST RESEARCH & TECHNOLOGY DEUTSCHLAND GMBH & CO. KG (DE) 1998-01-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120165369-A1 3-SUBSTITUTED QUINOLINIUM AND 7H-INDOLO[2,3-c]QUINOLINIUM SALTS AS NEW ANTIINFECTIVES IDO1, IDO2, NQO2 KMT2A 2440/4885NPC1 3157/4885RAB9A 2825/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.