SCHEMBL8574591

SCHEMBL8574591

COc1ccc(-c2noc(Br)c2C)cc1

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.58
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
MAPT P10636 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
PTGS1 P23219 1/20 0.44
PDE3A Q14432 1/20 0.44
NR1H4 Q96RI1 2/20 0.44
S1PR1 P21453 1/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
NFKB1 P19838 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5729316 0.81 PTGS2 (0.60) PTGS2NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL5730934 0.76 PTGS2 (0.54) PTGS2NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL28805031 0.74 PTGS2 (0.53) PTGS2MAPTPTGS1PDE3A
SCHEMBL2760349 0.74 PTGS2 (1.00) PTGS2PTGS1PDE3A
SCHEMBL5585925 0.72 ALDH1A1 (0.46) PTGS2NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL12987691 0.71 PTGS2 (0.56) PTGS2NPSR1MEN1KMT2A
SCHEMBL2776545 0.70 TARBP2 (0.54) PTGS2NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL5729672 0.70 PTGS2 (0.70) PTGS2PTGS1PDE3A
SCHEMBL4221887 0.70 MEN1 (0.55) PTGS2RAB9ANPSR1MEN1KMT2A
SCHEMBL4029497 0.70 PTGS2 (0.64) PTGS2NPC1RAB9ASMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998015541-A1 NOVEL ISOXAZOL DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME, AND A PROCESS FOR THE PREPARATION OF THE NOVEL COMPOUNDS EGIS Gyógyszergyár Rt. (HU) 1998-04-16 WO disclosed