SCHEMBL8575206

SCHEMBL8575206

CC(O)Cc1ccc(C#N)c(N)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 4/20 0.41
CYP3A4 P08684 3/20 0.41
TSHR P16473 2/20 0.41
CYP1A2 P05177 2/20 0.41
ADRB2 P07550 1/20 0.41
ADRB1 P08588 1/20 0.41
ADRB3 P13945 1/20 0.41
KDM4E B2RXH2 3/20 0.34
ALDH1A1 P00352 3/20 0.34
USP2 O75604 2/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
SLC22A12 Q96S37 1/20 0.34
ALOX15 P16050 3/20 0.33
ALOX12 P18054 3/20 0.33
MEN1 O00255 2/20 0.33
ESR1 P03372 2/20 0.33
TP53 P04637 2/20 0.33
HPGD P15428 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1931120 0.81 SLC22A12 (0.51) MAPK1CYP3A4TSHRCYP1A2ADRB2
SCHEMBL18930745 0.79 PRKACA (0.40) MAPK1CYP3A4TSHRCYP1A2ADRB2
SCHEMBL2371118 0.78 ALOX15 (0.39) MAPK1CYP3A4CYP1A2KDM4EALDH1A1
SCHEMBL29634742 0.78 ALOX15 (0.39) MAPK1CYP3A4CYP1A2KDM4EALDH1A1
SCHEMBL286459 0.78 AR (0.51) KDM4EALDH1A1USP2ALOX15ALOX12
Hydrochloric Acid SCHEMBL21144975 0.78 PRKACA (0.40) MAPK1CYP3A4TSHRCYP1A2ADRB2
Hydrochloric Acid SCHEMBL21144976 0.78 PRKACA (0.40) MAPK1CYP3A4TSHRCYP1A2ADRB2
SCHEMBL10971792 0.77 CYP2A6 (0.47) CYP3A4TSHRCYP1A2KDM4EALDH1A1
SCHEMBL22939708 0.76 GAA (0.44) CYP3A4TSHRKDM4EALDH1A1USP2
SCHEMBL1908021 0.75 TRPA1 (0.38) MAPK1CYP3A4TSHRCYP1A2ADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5852192-A Cyclic urea derivatives, pharmaceutical compositions containing these compounds and processes for preparing them DR. KARL THOMAE GMBH (DE) 1998-12-22 US disclosed