SCHEMBL8575481

SCHEMBL8575481

CSC(NCc1cccc(CNC(=O)OC(C)(C)C)c1)=C(C#N)C#N

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GLS O94925 5/20 0.48
CTSS P25774 7/20 0.41
CTSK P43235 5/20 0.41
CTSB P07858 3/20 0.41
BRD4 O60885 3/20 0.41
NAMPT P43490 2/20 0.41
CTSL P07711 2/20 0.41
CREBBP Q92793 1/20 0.41
KDM4A O75164 1/20 0.40
IDO1 P14902 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8579767 0.90 NAMPT (0.46) CTSSCTSKNAMPT
SCHEMBL8579008 0.89 AURKA (0.46) GLSCTSSCTSKCTSBBRD4
SCHEMBL6187053 0.89 BRD4 (0.45) GLSCTSSCTSKCTSBBRD4
SCHEMBL8605367 0.86 KCNA5 (0.43) CTSSCTSKCTSBNAMPTCTSL
SCHEMBL6186560 0.82 NAMPT (0.52) NAMPT
SCHEMBL24087990 0.80 GLS (0.51) GLSCTSSCTSKCTSBBRD4
SCHEMBL16181822 0.80 GLS (0.55) GLSCTSSCTSKCTSBBRD4
SCHEMBL352314 0.78 ERCC1 (0.52) GLSCTSSCTSKCTSBBRD4
SCHEMBL6187094 0.77 TDP1 (0.44) CTSSCTSKCTSBCTSLIDO1
SCHEMBL1165088 0.77 GLS (0.55) GLSBRD4NAMPTCREBBPKDM4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998014449-A1 FUSED PYRAZOLE DERIVATIVES AND PROCESSES FOR THEIR PREPARATION NOVARTIS AG (CH) 1998-04-09 WO disclosed