SCHEMBL8605367

SCHEMBL8605367

CSC(NCc1ccccc1CNC(=O)OC(C)(C)C)=C(C#N)C#N

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 1/20 0.43
KDM4A O75164 1/20 0.42
CTSS P25774 10/20 0.41
CTSK P43235 7/20 0.41
NAMPT P43490 1/20 0.40
CTSL P07711 2/20 0.40
CTSB P07858 2/20 0.40
IDO1 P14902 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
BCHE P06276 1/20 0.37
NQO2 P16083 1/20 0.37
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA7 P43166 1/20 0.36
CA14 Q9ULX7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8579767 0.88 NAMPT (0.46) CTSSCTSKNAMPTCA1
SCHEMBL8575481 0.86 GLS (0.48) KDM4ACTSSCTSKNAMPTCTSL
SCHEMBL30159605 0.81 KCNA5 (0.56) KCNA5KDM4ACTSSCTSKNAMPT
SCHEMBL8018113 0.81 KCNA5 (0.56) KCNA5KDM4ACTSSCTSKNAMPT
SCHEMBL6186560 0.80 NAMPT (0.52) NAMPTHDAC6
SCHEMBL6320846 0.79 KCNA5 (0.51) KCNA5KDM4ACTSSCTSKNAMPT
SCHEMBL6187094 0.79 TDP1 (0.44) CTSSCTSKCTSLCTSBIDO1
SCHEMBL8579008 0.78 AURKA (0.46) CTSSCTSKNAMPTCTSLCTSB
SCHEMBL6187053 0.78 BRD4 (0.45) CTSSCTSKNAMPTCTSBCA1
SCHEMBL5855817 0.77 KCNA5 (0.48) KCNA5KDM4ACTSSCTSKNAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998014449-A1 FUSED PYRAZOLE DERIVATIVES AND PROCESSES FOR THEIR PREPARATION NOVARTIS AG (CH) 1998-04-09 WO disclosed