SCHEMBL8575536

SCHEMBL8575536

O=C1c2c(O)cc(O)cc2OCC1(c1ccccc1)c1cccc(Br)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.37
CYP1A1 P04798 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP1B1 Q16678 1/20 0.37
MEN1 O00255 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
MAPT P10636 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
KMT2A Q03164 1/20 0.37
HSD17B10 Q99714 1/20 0.37
PNLIP P16233 1/20 0.35
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
HCAR3 P49019 1/20 0.34
HCAR2 Q8TDS4 1/20 0.34
ABCC2 Q92887 1/20 0.34
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8577523 0.88 ABCG2 (0.42) CYP19A1CYP3A4MAPTCYP2C9CYP2C19
SCHEMBL8574474 0.86 PLK1 (0.37) HCAR3HCAR2OPRM1OPRD1ALDH1A1
SCHEMBL8572826 0.86 CYP19A1 (0.37) CYP19A1CYP1A1CYP1A2CYP1B1MEN1
SCHEMBL8576046 0.80 HCAR3 (0.32) CYP3A4MAPTHCAR3HCAR2ALDH1A1
SCHEMBL8576216 0.79 GAA (0.38) MEN1MAPTKMT2AHCAR3HCAR2
SCHEMBL8577388 0.78 GAA (0.39) CYP1A2MEN1MAPTCYP2C19KMT2A
SCHEMBL571667 0.75 CYP19A1 (0.41) CYP19A1CYP1A1CYP1A2CYP1B1MEN1
SCHEMBL8577569 0.75 ABCG2 (0.42) CYP19A1CYP3A4MAPTCYP2C9CYP2C19
SCHEMBL28636154 0.72 MAPT (0.39) CYP19A1CYP1A1CYP1A2CYP1B1MEN1
SCHEMBL8572760 0.72 PLK1 (0.37) MAOAHCAR3HCAR2ALDH1A1HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998017662-A1 PHENYL-SUBSTITUTED BICYCLIC HETEROCYCLYL DERIVATIVES AND THEIR USE NOVARTIS AG (CH) 1998-04-30 WO claimed
WO-1998017662-A1 PHENYL-SUBSTITUTED BICYCLIC HETEROCYCLYL DERIVATIVES AND THEIR USE NOVARTIS AG (CH) 1998-04-30 WO disclosed