SCHEMBL8575938

SCHEMBL8575938

Cc1c(N2CCCC(C)(N)C2)c(F)cn2c(=O)c(C(=O)O)cc(C3CC3)c12

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SCN5A Q14524 1/20 0.42
KCNH2 Q12809 6/20 0.38
DPP4 P27487 7/20 0.33
CYP3A4 P08684 4/20 0.33
CYP2D6 P10635 3/20 0.32
PIM2 Q9P1W9 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
SCN9A Q15858 2/20 0.31
HPGD P15428 1/20 0.31
HSD17B10 Q99714 1/20 0.31
CYP1A2 P05177 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7499392 0.99 SCN5A (0.42) SCN5AKCNH2DPP4CYP3A4CYP2D6
SCHEMBL8570477 0.95 SCN5A (0.45) SCN5AKCNH2KDM4EALDH1A1
Hydrochloric Acid SCHEMBL7496978 0.94 SCN5A (0.45) SCN5AKCNH2KDM4EALDH1A1HPGD
SCHEMBL7508971 0.87 SCN5A (0.34) SCN5AKCNH2DPP4CYP3A4CYP2D6
SCHEMBL14515902 0.87 SCN5A (0.40) SCN5AKCNH2KDM4EALDH1A1HPGD
SCHEMBL8565903 0.86 SCN5A (0.44) SCN5AKCNH2KDM4EALDH1A1
SCHEMBL7927938 0.86 SCN5A (0.44) SCN5AKCNH2ALDH1A1
Hydrochloric Acid SCHEMBL9055075 0.85 SCN5A (0.43) SCN5AKCNH2KDM4EALDH1A1HPGD
Hydrochloric Acid SCHEMBL8573819 0.85 SCN5A (0.44) SCN5AKCNH2KDM4EALDH1A1
SCHEMBL8563910 0.85 SCN5A (0.44) SCN5AKCNH2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5599816-A BACTERICIDE ABBOTT LABORATORIES (US) 1997-02-04 US claimed
WO-1996039407-A1 QUINOLIZINONE TYPE COMPOUNDS ABBOTT LABORATORIES (US) 1996-12-12 WO claimed
US-5726182-A TREATMENT OF BACTERIAL INFECTIONS ABBOTT LABORATORIES (US) 1998-03-10 US disclosed
US-5599816-A BACTERICIDE ABBOTT LABORATORIES (US) 1997-02-04 US disclosed
WO-1996039407-A1 QUINOLIZINONE TYPE COMPOUNDS ABBOTT LABORATORIES (US) 1996-12-12 WO disclosed