SCHEMBL8575969

SCHEMBL8575969

CCCCOc1cc(C2CN(C)C(=O)N2)ccc1OC

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 11/20 0.57
PDE4B Q07343 10/20 0.57
PDE4D Q08499 7/20 0.57
PDE4C Q08493 6/20 0.57
MAPK1 P28482 2/20 0.49
LMNA P02545 2/20 0.49
TNF P01375 1/20 0.49
MAPT P10636 1/20 0.49
PDE3B Q13370 1/20 0.49
PDE3A Q14432 1/20 0.49
KDM4E B2RXH2 1/20 0.49
MEN1 O00255 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
NFKB1 P19838 1/20 0.49
KMT2A Q03164 1/20 0.49
TP53 P04637 1/20 0.41
GAA P10253 1/20 0.41
HTR2C P28335 1/20 0.41
GFER P55789 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2779051 0.80 PDE4A (0.65) PDE4APDE4BPDE4DPDE4CMAPK1
SCHEMBL8575965 0.76 PDE4A (0.63) PDE4APDE4BPDE4DPDE4CMAPK1
SCHEMBL6584261 0.74 PDE4B (0.51) PDE4APDE4BPDE4DPDE4CMAPK1
SCHEMBL5324227 0.72 PDE4A (1.00) PDE4APDE4BPDE4DPDE4CMAPK1
SCHEMBL11427405 0.72 PDE4A (0.64) PDE4APDE4BPDE4DPDE4CMAPK1
SCHEMBL2779053 0.71 PDE4A (0.51) PDE4APDE4BPDE4DPDE4CMAPK1
SCHEMBL6232676 0.71 PDE4A (0.54) PDE4APDE4BPDE4DPDE4CMAPK1
SCHEMBL6587870 0.71 PDE4A (0.58) PDE4APDE4BPDE4DPDE4CMAPK1
SCHEMBL7913434 0.70 PDE4A (0.67) PDE4APDE4BPDE4DPDE4CMAPK1
SCHEMBL6232341 0.70 PDE4A (0.60) PDE4APDE4BPDE4DPDE4CMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117241803-A Purine nucleosides, intermediates and methods of making the same 阿斯特罗赛特制药公司 2023-12-15 CN disclosed
CN-110003212-B A3 adenosine receptor agonists 美国卫生和人力服务部 2022-12-06 CN disclosed
US-5849774-A Treatment of sepsis-induced acute renal failure UNIVERSITY OF PITTSBURGH (US) 1998-12-15 US disclosed