SCHEMBL8577314

SCHEMBL8577314

N#Cc1cc(F)cc(C(=O)N2CCNCC2)c1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SCN5A Q14524 3/20 0.49
SCN9A Q15858 3/20 0.49
SIGMAR1 Q99720 1/20 0.47
GRM5 P41594 4/20 0.46
PKM P14618 1/20 0.43
ALDH1A1 P00352 1/20 0.43
TDO2 P48775 1/20 0.43
USP2 O75604 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
HPGD P15428 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1934997 0.88 SCN5A (0.51) SCN5ASCN9AGRM5ALDH1A1USP2
SCHEMBL2740504 0.78 SIGMAR1 (0.61) SIGMAR1GRM5ALDH1A1USP2CYP3A4
SCHEMBL19404236 0.78 CTNNB1 (0.53) SIGMAR1
Hydrochloric Acid SCHEMBL223669 0.77 SIGMAR1 (0.59) SIGMAR1GRM5ALDH1A1USP2CYP3A4
SCHEMBL1375337 0.76 SIGMAR1 (0.64) SCN9ASIGMAR1ALDH1A1CYP3A4HPGD
SCHEMBL851451 0.76 SCN9A (0.63) SCN9ASIGMAR1CYP3A4
Hydrochloric Acid SCHEMBL7718789 0.75 SIGMAR1 (0.62) SCN9ASIGMAR1ALDH1A1CYP3A4HPGD
SCHEMBL226167 0.74 SIGMAR1 (0.56) SIGMAR1PKMTDO2HPGD
SCHEMBL2336862 0.74 SMN1; SMN2 (0.71) SIGMAR1ALDH1A1USP2CYP3A4HPGD
SCHEMBL24088883 0.73 GABRD (0.52) SIGMAR1PKMTDO2USP2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012068450-A1 CYCLOBUTYL SUBSTITUTED PYRROLOPYRIDINE AND PYRROLOPYRIMIDINE DERIVATIVES AS JAK INHIBITORS INCYTE CORPORATION (US) 2012-05-24 WO disclosed