SCHEMBL8577758

SCHEMBL8577758

O=C(O)NCC(O)C(CC1CCCCC1)NC(=O)O

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.41
PSEN1 P49768 1/20 0.38
PSEN2 P49810 1/20 0.38
APH1B Q8WW43 1/20 0.38
NCSTN Q92542 1/20 0.38
APH1A Q96BI3 1/20 0.38
PSENEN Q9NZ42 1/20 0.38
REN P00797 4/20 0.38
BCHE P06276 3/20 0.36
LTA4H P09960 1/20 0.35
GRN P28799 1/20 0.35
SORT1 Q99523 1/20 0.35
CTSK P43235 3/20 0.35
CTSS P25774 2/20 0.35
METAP2 P50579 2/20 0.35
METAP1 P53582 1/20 0.35
CTSL P07711 1/20 0.34
CTSB P07858 1/20 0.34
CPB2 Q96IY4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7312864 0.89 PSEN1 (0.38) CYP2D6PSEN1PSEN2APH1BNCSTN
SCHEMBL970762 0.84 GRN (0.40) CYP2D6PSEN1PSEN2APH1BNCSTN
SCHEMBL969137 0.84 GRN (0.40) CYP2D6PSEN1PSEN2APH1BNCSTN
SCHEMBL967760 0.84 GRN (0.40) CYP2D6PSEN1PSEN2APH1BNCSTN
SCHEMBL3347419 0.84 PSEN1 (0.39) CYP2D6PSEN1PSEN2APH1BNCSTN
SCHEMBL4430800 0.83 CTSS (0.55) RENCTSKCTSS
SCHEMBL968972 0.83 CYP2D6 (0.42) CYP2D6PSEN1PSEN2APH1BNCSTN
SCHEMBL968973 0.83 CYP2D6 (0.42) CYP2D6PSEN1PSEN2APH1BNCSTN
SCHEMBL3382250 0.82 PSEN1 (0.37) CYP2D6PSEN1PSEN2APH1BNCSTN
SCHEMBL4433209 0.79 REN (0.50) CYP2D6RENBCHEMETAP2METAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776933-A Method of inhibiting protease E. R. SQUIBB & SONS, INC. (US) 1998-07-07 US disclosed
US-5760036-A ENZYME INHIBITORS OF RETROVIRAL PROTEASE FOR PREVENTION OF AIDS E. R. SQUIBB & SONS, INC. (US) 1998-06-02 US disclosed