SCHEMBL8577867

SCHEMBL8577867

CCCn1c(=O)c2c(nc(C3CCCC3)n2Cc2ccccc2)n(CCOC)c1=O

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 13/20 0.57
ADORA2A P29274 3/20 0.57
ADORA2B P29275 3/20 0.57
ADORA1 P30542 3/20 0.53
KMT2A Q03164 1/20 0.52
PDE5A O76074 2/20 0.50
DCTPP1 Q9H773 1/20 0.48
LMNA P02545 1/20 0.48
THRB P10828 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8576968 0.94 ADORA3 (0.56) ADORA3ADORA2AADORA2BADORA1KMT2A
SCHEMBL8577877 0.89 ADORA2B (0.60) ADORA3ADORA2AADORA2BADORA1KMT2A
SCHEMBL8576951 0.89 ADORA3 (0.61) ADORA3ADORA2AADORA2BADORA1KMT2A
SCHEMBL8576493 0.88 ADORA2A (0.59) ADORA3ADORA2AADORA2BADORA1KMT2A
SCHEMBL8576500 0.87 ADORA3 (0.58) ADORA3ADORA2AADORA2BADORA1KMT2A
SCHEMBL8579493 0.86 ADORA3 (0.60) ADORA3ADORA2AADORA2BADORA1KMT2A
SCHEMBL8576828 0.86 ADORA3 (0.57) ADORA3ADORA2AADORA2BADORA1KMT2A
SCHEMBL8579688 0.86 ADORA3 (0.60) ADORA3ADORA2AADORA2BADORA1KMT2A
SCHEMBL8578138 0.86 ADORA3 (0.56) ADORA3ADORA2AADORA2BADORA1KMT2A
SCHEMBL8579260 0.86 ADORA3 (0.56) ADORA3ADORA2AADORA2BADORA1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719279-A CHOLINOMIMETICS BOEHRINGER INGELHEIM KG (DE) 1998-02-17 US disclosed
WO-1994003456-A1 ASYMMETRICALLY SUBSTITUTED XANTHINE WITH ADENOSINE-ANTAGONISTIC PROPERTIES BOEHRINGER INGELHEIM KG (DE) 1994-02-17 WO disclosed