SCHEMBL8580592

SCHEMBL8580592

CC(=O)Nc1c(C(=O)O)ccc(F)c1F

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 3/20 0.50
MAP2K2 P36507 2/20 0.50
KDM4E B2RXH2 4/20 0.44
HSD17B10 Q99714 2/20 0.44
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.39
NAPRT Q6XQN6 1/20 0.38
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
GRIK1 P39086 1/20 0.37
MAPK1 P28482 1/20 0.37
ALDH1A1 P00352 1/20 0.36
MYC P01106 1/20 0.36
CYP1A2 P05177 1/20 0.35
HDAC1 Q13547 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30956704 0.86 KDM4E (0.44) MAP2K1MAP2K2KDM4EHSD17B10CES2
SCHEMBL20819607 0.86 KDM4E (0.44) MAP2K1MAP2K2KDM4EHSD17B10CES2
SCHEMBL29181923 0.83 RXFP1 (0.39) MAP2K1MAP2K2KDM4EHSD17B10SMN1; SMN2
SCHEMBL28091550 0.79 KDM4E (0.40) MAP2K1MAP2K2KDM4EHSD17B10SMN1; SMN2
SCHEMBL16075172 0.78 ALDH1A1 (0.47) HSD17B10CES2CES1SMN1; SMN2NAPRT
SCHEMBL2892368 0.78 MAOA (0.42) KDM4EHSD17B10SMN1; SMN2MEN1KMT2A
SCHEMBL22642784 0.76 HDAC1 (0.48) SMN1; SMN2MEN1KMT2AALDH1A1HDAC1
SCHEMBL21807214 0.76 RXFP1 (0.42) HSD17B10CES2CES1SMN1; SMN2NAPRT
SCHEMBL670931 0.76 KDM4E (0.45) MAP2K1KDM4EHSD17B10SMN1; SMN2MEN1
SCHEMBL7554525 0.76 MAP2K1 (0.48) MAP2K1MAP2K2KDM4EHSD17B10CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998011438-A1 SYNTHESIS OF QUINAZOLINONE LIBRARIES AND DERIVATIVES THEREOF TREGA BIOSCIENCES, INC. (US) 1998-03-19 WO disclosed