SCHEMBL8581793

SCHEMBL8581793

O=c1[nH]c(=O)n(CCc2ccc(Cl)cc2)c2nc(C3CCCC3)n(Cc3ccccc3)c12

nearest known ligand 0.66

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 8/20 0.66
MEN1 O00255 7/20 0.49
POLB P06746 2/20 0.49
RAB9A P51151 1/20 0.49
TSHR P16473 7/20 0.47
NPSR1 Q6W5P4 2/20 0.47
ALDH1A1 P00352 8/20 0.46
HTT P42858 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
USP2 O75604 2/20 0.46
ATM Q13315 1/20 0.45
APOBEC3G Q9HC16 1/20 0.45
MAPK1 P28482 2/20 0.45
HPGD P15428 1/20 0.44
HSD17B10 Q99714 1/20 0.44
BRAF P15056 1/20 0.44
MAPT P10636 1/20 0.44
ADORA3 P0DMS8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8576721 0.89 KMT2A (0.64) KMT2AMEN1POLBRAB9ATSHR
SCHEMBL9168640 0.86 KMT2A (0.74) KMT2AMEN1POLBRAB9ATSHR
SCHEMBL8579681 0.83 KMT2A (0.62) KMT2AMEN1POLBRAB9ATSHR
SCHEMBL8577929 0.83 KMT2A (0.70) KMT2AMEN1POLBRAB9ATSHR
SCHEMBL8576289 0.82 ADORA3 (0.56) KMT2AADORA3
SCHEMBL9708443 0.82 KMT2A (0.55) KMT2AMEN1POLBRAB9ATSHR
SCHEMBL8581812 0.82 KMT2A (0.67) KMT2AMEN1POLBRAB9ATSHR
SCHEMBL6094064 0.81 KMT2A (0.70) KMT2AMEN1POLBRAB9ATSHR
SCHEMBL8606081 0.79 KMT2A (0.66) KMT2AMEN1POLBRAB9ATSHR
SCHEMBL27523019 0.79 KMT2A (0.63) KMT2AMEN1POLBRAB9ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1043348-C Asymmetrically substituted xanthines BOEHRINGER INGELHEIM KG (DE) 1999-05-12 CN disclosed
US-5719279-A CHOLINOMIMETICS BOEHRINGER INGELHEIM KG (DE) 1998-02-17 US disclosed
WO-1994003456-A1 ASYMMETRICALLY SUBSTITUTED XANTHINE WITH ADENOSINE-ANTAGONISTIC PROPERTIES BOEHRINGER INGELHEIM KG (DE) 1994-02-17 WO disclosed