SCHEMBL8577929

SCHEMBL8577929

COCCn1c(=O)[nH]c(=O)c2c1nc(C1CCCC1)n2Cc1ccccc1

nearest known ligand 0.70

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 7/20 0.70
ALDH1A1 P00352 9/20 0.56
KDM4E B2RXH2 6/20 0.56
PKM P14618 2/20 0.56
MAPK1 P28482 2/20 0.53
GAA P10253 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
RECQL P46063 1/20 0.53
MEN1 O00255 6/20 0.52
POLB P06746 1/20 0.52
RAB9A P51151 1/20 0.52
HPGD P15428 4/20 0.51
HSD17B10 Q99714 1/20 0.51
NPSR1 Q6W5P4 4/20 0.50
TSHR P16473 2/20 0.50
HTT P42858 4/20 0.49
MAPT P10636 2/20 0.49
BRAF P15056 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8581812 0.94 KMT2A (0.67) KMT2AALDH1A1KDM4EPKMMAPK1
SCHEMBL9168640 0.89 KMT2A (0.74) KMT2AALDH1A1KDM4EMAPK1SMN1; SMN2
SCHEMBL6094064 0.86 KMT2A (0.70) KMT2AALDH1A1KDM4EPKMMAPK1
SCHEMBL8576721 0.86 KMT2A (0.64) KMT2AALDH1A1KDM4EMAPK1GAA
SCHEMBL8606081 0.86 KMT2A (0.66) KMT2AALDH1A1KDM4EMAPK1GAA
SCHEMBL27523019 0.85 KMT2A (0.63) KMT2AALDH1A1KDM4EPKMMAPK1
SCHEMBL8579681 0.84 KMT2A (0.62) KMT2AALDH1A1KDM4EMAPK1GAA
SCHEMBL9707780 0.84 KMT2A (0.53) KMT2AALDH1A1KDM4EPKMMAPK1
SCHEMBL8581793 0.83 KMT2A (0.66) KMT2AALDH1A1MAPK1SMN1; SMN2MEN1
SCHEMBL8577867 0.82 ADORA3 (0.57) KMT2ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1043348-C Asymmetrically substituted xanthines BOEHRINGER INGELHEIM KG (DE) 1999-05-12 CN disclosed
US-5719279-A CHOLINOMIMETICS BOEHRINGER INGELHEIM KG (DE) 1998-02-17 US disclosed
EP-0654033-A1 ASYMMETRICALLY SUBSTITUTED XANTHINE WITH ADENOSINE-ANTAGONISTIC PROPERTIES BOEHRINGER INGELHEIM KG (DE) 1995-05-24 EP disclosed
WO-1994003456-A1 ASYMMETRICALLY SUBSTITUTED XANTHINE WITH ADENOSINE-ANTAGONISTIC PROPERTIES BOEHRINGER INGELHEIM KG (DE) 1994-02-17 WO disclosed