SCHEMBL8583399

SCHEMBL8583399

CCOC(=O)C[C@H](NO)C(=O)OCC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.50
MGAM O43451 1/20 0.50
SI P14410 1/20 0.50
MGAM2 Q2M2H8 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.49
KMT2A Q03164 2/20 0.46
POLB P06746 1/20 0.46
ALDH1A1 P00352 6/20 0.42
CYP3A4 P08684 2/20 0.42
ALOX15 P16050 2/20 0.42
TSHR P16473 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
TRPA1 O75762 1/20 0.41
HSD17B10 Q99714 2/20 0.41
CHRM1 P11229 1/20 0.41
ADORA1 P30542 1/20 0.41
CAD P27708 1/20 0.41
CYP1A2 P05177 2/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8583393 1.00 GAA (0.50) GAAMGAMSIMGAM2L3MBTL1
SCHEMBL15257970 0.84 GAA (0.46) GAAMGAMSIMGAM2L3MBTL1
SCHEMBL13624780 0.83 GAA (0.50) GAAMGAMSIMGAM2L3MBTL1
SCHEMBL25274352 0.82 CAD (0.47) GAAMGAMSIMGAM2L3MBTL1
SCHEMBL10612838 0.82 GAA (0.48) GAAMGAMSIMGAM2L3MBTL1
SCHEMBL9729395 0.82 GAA (0.48) GAAMGAMSIMGAM2L3MBTL1
SCHEMBL8583427 0.80 L3MBTL1 (0.36) GAAMGAMSIMGAM2L3MBTL1
SCHEMBL8583430 0.80 L3MBTL1 (0.36) GAAMGAMSIMGAM2L3MBTL1
SCHEMBL468760 0.80 L3MBTL1 (0.50) GAAMGAMSIMGAM2L3MBTL1
SCHEMBL3565347 0.80 L3MBTL1 (0.69) GAAMGAMSIMGAM2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5405987-A N-hydroxyaspartic acid derivatives; chemical intermediates HOECHST CELANESE CORPORATION (US) 1995-04-11 US claimed
US-5322948-A Reacting unsaturated diacid or derivative with hydroxylamine or a salt thereof to form N-hydroxy-2-aminobutane diacid derivative HOECHST CELANESE CORPORATION (US) 1994-06-21 US claimed
EP-0511446-A2 Process for preparing pyridinecarboxylic acid derivatives HOECHST CELANESE CORPORATION (US) 1992-11-04 EP claimed
CN-1058205-A The method for preparing pyridine and quinoline HOECHST CELANESE CORP (US) 1992-01-29 CN claimed
EP-0452094-A2 A method of the preparation of N-hydroxy aspartic acid derivate HOECHST CELANESE CORPORATION (US) 1991-10-16 EP claimed
CN-1049844-A The preparation method of pyridine carboxylic acid derivatives HOECHST CELANESE CORP (US) 1991-03-13 CN claimed
EP-0415767-A2 Process for preparing pyridine carboxylic acid derivatives HOECHST CELANESE CORPORATION (US) 1991-03-06 EP claimed
US-5808067-A Process for preparing pyridine and quinoline derivatives HOECHST CELANESE CORPORATION (US) 1998-09-15 US disclosed
US-5405987-A N-hydroxyaspartic acid derivatives; chemical intermediates HOECHST CELANESE CORPORATION (US) 1995-04-11 US disclosed
US-5322948-A Reacting unsaturated diacid or derivative with hydroxylamine or a salt thereof to form N-hydroxy-2-aminobutane diacid derivative HOECHST CELANESE CORPORATION (US) 1994-06-21 US disclosed
EP-0564083-A1 Conversion of pyridine-2,3-dicarboxylic acid esters to their cyclic anhydrides HOECHST CELANESE CORPORATION (US) 1993-10-06 EP disclosed
US-5208342-A Hydrolysis and dehydration HOECHST CELANESE CORPORATION (US) 1993-05-04 US disclosed
EP-0511446-A2 Process for preparing pyridinecarboxylic acid derivatives HOECHST CELANESE CORPORATION (US) 1992-11-04 EP disclosed
CN-1058205-A The method for preparing pyridine and quinoline HOECHST CELANESE CORP (US) 1992-01-29 CN disclosed
EP-0452094-A2 A method of the preparation of N-hydroxy aspartic acid derivate HOECHST CELANESE CORPORATION (US) 1991-10-16 EP disclosed
CN-1049844-A The preparation method of pyridine carboxylic acid derivatives HOECHST CELANESE CORP (US) 1991-03-13 CN disclosed
EP-0415767-A2 Process for preparing pyridine carboxylic acid derivatives HOECHST CELANESE CORPORATION (US) 1991-03-06 EP disclosed