SCHEMBL858532

SCHEMBL858532

CCc1ccc(CNCc2[nH]c3ncccc3c2-c2ccc(C(N)=O)cc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CAMKK2 Q96RR4 4/20 0.45
RIPK1 Q13546 1/20 0.42
CHUK O15111 4/20 0.41
INSR P06213 3/20 0.41
MAPK8 P45983 3/20 0.41
ALDH1A1 P00352 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MKNK1 Q9BUB5 2/20 0.39
MKNK2 Q9HBH9 2/20 0.39
CHEK2 O96017 4/20 0.38
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37
OPRK1 P41145 1/20 0.37
AURKA O14965 1/20 0.36
RPS6KB1 P23443 1/20 0.36
IKBKB O14920 1/20 0.36
TRPV1 Q8NER1 1/20 0.36
HDAC1 Q13547 2/20 0.36
HDAC3 O15379 1/20 0.36
ERBB2 P04626 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14620968 0.90 CAMKK2 (0.46) CAMKK2RIPK1CHUKINSRMAPK8
SCHEMBL7985889 0.89 VNN1 (0.46) CAMKK2RIPK1CHUKINSRMAPK8
SCHEMBL858803 0.81 CAMKK2 (0.44) CAMKK2RIPK1CHUKINSRMAPK8
SCHEMBL15298804 0.75 CAMKK2 (0.43) CAMKK2RIPK1CHUKINSRMAPK8
SCHEMBL857545 0.75 CAMKK2 (0.47) CAMKK2RIPK1CHUKINSRMAPK8
SCHEMBL858429 0.74 MAPK14 (0.52) ALDH1A1NPSR1
SCHEMBL20086210 0.73 CA1 (0.50) ALDH1A1IKBKBKDR
SCHEMBL857420 0.73 MAPK13 (0.41)
SCHEMBL857332 0.73 CAMKK2 (0.46) CAMKK2RIPK1CHUKINSRMAPK8
SCHEMBL14620869 0.73 CAMKK2 (0.42) CAMKK2RIPK1CHUKINSRMAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143271-B2 Compounds and methods for kinase modulation, and indications therefor PLEXXIKON INC. (US) 2012-03-27 US disclosed