SCHEMBL8586471

SCHEMBL8586471

NCCc1csc2cccc(O)c12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.49
TAAR1 Q96RJ0 4/20 0.48
CYP2A6 P11509 2/20 0.42
CA2 P00918 2/20 0.39
MEN1 O00255 2/20 0.37
RAD52 P43351 2/20 0.37
RECQL P46063 2/20 0.37
KMT2A Q03164 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
GAPDH P04406 1/20 0.37
THRB P10828 1/20 0.37
APEX1 P27695 1/20 0.37
BLM P54132 1/20 0.37
HMGB1 P09429 1/20 0.37
KDM4E B2RXH2 1/20 0.36
MAPT P10636 1/20 0.36
ALOX15 P16050 1/20 0.36
MAPK1 P28482 1/20 0.36
HSD17B10 Q99714 1/20 0.36
AGO2 Q9UKV8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8587901 0.81 HTR2A (0.47) HTR2CTAAR1CYP2A6CA2KDM4E
SCHEMBL1727943 0.80 CYP2A6 (0.43) CYP2A6CA2KDM4E
SCHEMBL8585665 0.79 CA2 (0.56) HTR2CTAAR1CYP2A6CA2ALDH1A1
SCHEMBL8584219 0.79 TAAR1 (0.50) TAAR1CYP2A6CA2DRD2
SCHEMBL25030243 0.79 HTR2A (0.54) HTR2CTAAR1CYP2A6CA2MEN1
SCHEMBL25028212 0.79 HTR2A (0.58) HTR2CCYP2A6DRD1ALDH1A1CYP1A2
SCHEMBL25029525 0.76 HTR2A (0.39) CYP2A6CA2ALDH1A1CYP1A2CYP2D6
SCHEMBL25029542 0.76 MPO (0.38) CYP2A6CA2ALDH1A1CYP1A2CYP2D6
SCHEMBL1727525 0.76 TP53 (0.42) HTR2CTAAR1CYP2A6CA2MAPT
SCHEMBL8586513 0.76 TAAR1 (0.53) TAAR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998027984-A1 METHOD OF PRODUCING ANALGESIA BY ADMINISTRATION OF 1,2,3,4-TETRAHYDROBENZO-[b]THIENO[2,3-c]PYRIDINE AND DERIVATIVES NEUREX CORPORATION (US) 1998-07-02 WO disclosed
US-4971974-A ANOREXIGENIC AGENTS, BENZO B!THIENO 2,3-C!PYRIDINE COMPOUNDS NEUREX CORPORATION (US) 1990-11-20 US disclosed