SCHEMBL8587237

SCHEMBL8587237

C1CCN(CCC2CC2)C1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.50
CHRM5 P08912 1/20 0.44
ADRA2C P18825 1/20 0.44
HRH3 Q9Y5N1 1/20 0.43
CARM1 Q86X55 1/20 0.39
PRMT6 Q96LA8 1/20 0.39
PRMT8 Q9NR22 1/20 0.39
DRD2 P14416 1/20 0.37
DRD3 P35462 1/20 0.37
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10153844 0.97 CYP1A2 (0.54) CYP1A2CHRM5ADRA2CHRH3CARM1
SCHEMBL10949210 0.92 CHRM5 (0.54) CYP1A2CHRM5ADRA2CHRH3
SCHEMBL30340999 0.90 CHRM5 (0.58) CYP1A2CHRM5ADRA2CHRH3
SCHEMBL12945 0.90 CHRM5 (0.58) CYP1A2CHRM5ADRA2CHRH3
SCHEMBL3218288 0.90 CHRM5 (0.58) CYP1A2CHRM5ADRA2CHRH3
SCHEMBL14686114 0.89 DRD2 (0.48) CYP1A2CHRM5ADRA2CHRH3DRD2
SCHEMBL14686115 0.89 DRD2 (0.48) CYP1A2CHRM5ADRA2CHRH3DRD2
Hydrochloric Acid SCHEMBL2514759 0.87 DRD2 (0.47) CYP1A2CHRM5ADRA2CHRH3DRD2
Hydrochloric Acid SCHEMBL2514757 0.87 DRD2 (0.47) CYP1A2CHRM5ADRA2CHRH3DRD2
SCHEMBL3437028 0.85 CYP1A2 (0.48) CYP1A2CHRM5ADRA2CHRH3CARM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108727343-A Quinazolinones PARP-1/2 inhibitor containing 3- amino nafoxidines and preparation method thereof, pharmaceutical composition and purposes 中国医学科学院药物研究所 2018-11-02 CN disclosed
WO-1998039295-A1 (R)N-(1-CYCLOPROPYLMETHYLPYRROLIDIN-2-YLMETHYL)BENZAMIDE AND ITS USE AS AN ANTIDIARRHOEAL JOUVEINAL (FR) 1998-09-11 WO disclosed